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(4aS,8aR)-1-(3-aminopropyl)-6-[(5-fluoro-2-methoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
2-cyclopropyl-9-{2-[ethyl(methyl)amino]acetyl}-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
5-({3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[4-({4-[3-(dimethylamino)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-4-amine
1-(2-ethylpyrimidine-5-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-2-methyl-1,3-thiazole-4-carboxamide
{4-[(2-chlorophenyl)methyl]-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}methanol
4-(3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-2,5-dimethyl-1H-pyrrol-1-yl)-4H-1,2,4-triazole
3,5-dimethyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
(3aS,6aS)-2-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[4-(4-methylbenzoyl)piperazin-1-yl]-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-[2-hydroxy-3-(4-methoxy-2-{[(2-methoxy-2-methylpropyl)amino]methyl}phenoxy)propyl]piperidin-4-ol
(3aS,6aS)-2-(3-chlorobenzoyl)-5-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{5-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
4-{[1-(4-fluorophenyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl]methyl}morpholine
1-(azocan-1-yl)-3-[5-({[(2,3-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
1'-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-1,2-dihydrospiro[indole-3,4'-piperidine]
1-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-3-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-5-yl)urea
5-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)pyrazine-2-carboxamide
3-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(2,6-dimethoxypyridin-3-yl)urea
{1-[(5-chlorothiophen-2-yl)sulfonyl]-4-(2-phenoxyethyl)piperidin-4-yl}methanol
({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)(cyclohexylmethyl)methylamine
2-{[4-(1-propyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
1-{[(3R,4R)-1-[1-(4-fluorophenyl)cyclopropanecarbonyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-1,2,3-thiadiazole-4-carboxamide
(2S,4S)-N,N-diethyl-4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
3-(2-hydroxypropan-2-yl)-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
3-{[3-(carboxymethyl)morpholin-4-yl]sulfonyl}-4-methoxybenzoic acid
3-(2-methoxyphenyl)-N-[(1-methylpyrrolidin-3-yl)methyl]benzamide
(1H-imidazol-2-ylmethyl)(prop-2-en-1-yl)(pyridin-2-ylmethyl)amine
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(1,3-thiazole-4-carbonyl)piperidine-3-carboxylate
1-{3-[2-(2,4,5-trimethylphenyl)-1H-imidazol-1-yl]propyl}-1H-1,2,4-triazole
4-(azocan-1-yl)-N-(1-methoxybutan-2-yl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
(1S,6R)-3-methyl-9-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-3-(3-fluorophenyl)propanamide
2-methyl-8-(2-phenylpropyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
ethyl 2-[1-(5-{[(5-chloropyridin-3-yl)oxy]methyl}-1,2-oxazole-3-amido)cyclohexyl]acetate
1-[(2,4-dimethoxyphenyl)methyl]-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
2-[2-(thiophen-2-yl)ethyl]-1-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidine
1-(cyclohexylmethyl)-5-(4-ethylpiperazine-1-carbonyl)piperidin-2-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-(pyridin-2-yl)propanamide
2-fluoro-N-[4-(4-{[(2-methylphenyl)(pyridin-4-yl)methyl]amino}piperidin-1-yl)phenyl]benzamide
1'-[(3-chloro-4-fluorophenyl)methyl]-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-[(2E)-2-methylbut-2-en-1-yl]-2,5-diazabicyclo[2.2.1]heptan-3-one
2-[(4-chlorophenyl)methyl]-8-(6-methoxypyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
9-[4-(1,3-oxazol-5-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-5-methyl-N-[2-(pyridin-4-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
3-cyclopentyl-1-[2-(1-ethylpiperidin-3-yl)ethyl]urea
9-(2,4-difluorophenyl)-15-methyl-12-(morpholine-4-carbonyl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one