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3-({[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amino)-N-(1,3-thiazol-2-yl)propanamide
3-({4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)-1,2-dihydroquinolin-2-one
N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)pyridine-2-carboxamide
(2S,4S)-4-amino-1-(4-methyl-5-phenylthiophene-2-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-{[(3-tert-butyl-1H-pyrazol-5-yl)methyl]sulfamoyl}-N,N-dimethylbenzamide
3-(2-oxo-2-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}ethyl)-1,3-oxazolidin-2-one
2-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-N-[(2-methylphenyl)methyl]acetamide
2-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-4-phenylazepane
N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
N-(prop-2-en-1-yl)-5-(quinolin-3-yl)furan-2-carboxamide
2-amino-N-({1-[(3-fluoropyridin-4-yl)methyl]pyrrolidin-3-yl}methyl)pyridine-4-carboxamide
5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-2-(pyridin-4-yl)pyridine
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(morpholin-3-yl)acetamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-methoxybenzamide
2-{5-[1-(dimethylcarbamoyl)piperidin-4-yl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
1-(1-{1-[4-(difluoromethoxy)benzoyl]piperidin-4-yl}ethyl)-4-methylpiperazine
4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-2-(4-fluorophenyl)morpholine
3-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
6-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-2-carboxylic acid
2-({2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}amino)-6-methyl-3,4-dihydropyrimidin-4-one
3-[(2-methyl-1,3-oxazol-4-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-(methoxymethyl)-N-[(2-methoxyphenyl)methyl]pyrimidin-4-amine
9-[2-(2-methylphenoxy)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-(4-methyl-1H-imidazole-5-carbonyl)piperidine
2-(3-methylbutyl)-8-[2-(2-oxopyrrolidin-1-yl)acetyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-methyl-7-[1-(propan-2-yl)piperidine-4-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
4-{[1-(3-fluorophenyl)-5-[2-(oxolan-2-yl)ethyl]-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
4-({1-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]pyrrolidin-3-yl}methyl)benzoic acid
8-cyclopentanecarbonyl-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
3-[({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]phenol
2-{[4-(oxan-2-ylmethyl)phenyl]sulfanyl}acetamide
N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-2,3-dimethyl-N-(pyridin-3-ylmethyl)-1H-indole-7-carboxamide
1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(4-fluorophenyl)methyl]-1,4-diazepane
5-(3-methoxyphenoxymethyl)-N-(3-methylbutyl)-1H-pyrazole-3-carboxamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-5-(2-methylphenyl)-1,2,4-triazin-3-amine
3-(2-{4-[(2,6,6-trimethylcyclohex-1-en-1-yl)methyl]-1H-1,2,3-triazol-1-yl}ethyl)-1,3-oxazolidin-2-one
3-[9-(2-ethoxyethyl)-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]propanamide
(3S,4S)-3,4-bis(hydroxymethyl)-N-[3-(3-methoxyphenyl)phenyl]pyrrolidine-1-carboxamide
methyl 1-{4-[ethyl(methyl)amino]pyrimidin-2-yl}piperidine-4-carboxylate
(1R,7S)-N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N-methyl-4-oxo-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-[4-({methyl[(1-methylpyrrolidin-2-yl)methyl]amino}methyl)-1H-pyrazol-1-yl]propanoic acid
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methoxypyrimidine-5-carboxamide
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
(2S,4R)-1-benzyl-4-(cyclooctylamino)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(isoquinolin-5-ylmethyl)-N-methyl-1-(oxan-4-yl)piperidine-3-carboxamide
(1R,3S)-3-methoxy-7-(2-methyl-6-propylpyrimidin-4-yl)-7-azaspiro[3.5]nonan-1-ol
2-[1-(1,3-thiazol-4-ylmethyl)pyrrolidin-2-yl]-1,3-thiazole