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1-[(3,5-dimethylphenyl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
N-(adamantan-1-yl)-2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]acetamide
3-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-1-(quinolin-6-yl)urea
4-(methoxymethyl)-6-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidine
1-(5-methyl-1,3-benzoxazol-2-yl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(3aR,6aR)-2-cyclopentyl-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-(azocan-1-yl)-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}propanamide
2-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
4-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-2-methylphenol
3-methoxy-1-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]propan-1-one
N-[(3R,4R)-3-hydroxy-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidin-4-yl]pyridine-2-carboxamide
{4-[(4-methoxyphenyl)methyl]-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl}methanol
3-[1-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)piperidin-3-yl]benzoic acid
(1S,5R)-6-(1H-pyrrole-2-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
6-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
1-(5-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)ethan-1-one
1-ethyl-5-[(4-hydroxyphenyl)methyl]-N-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(1-hydroxybutan-2-yl)-2,6-dimethyl-N-(pyridin-2-ylmethyl)quinoline-3-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-methylthieno[2,3-d]pyrimidin-4-amine
3-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-1-[3-(1H-1,2,3-triazol-1-yl)propyl]urea
2-[(4aR,7aS)-4-(1-methyl-1H-pyrrole-2-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
N-(3-hydroxypropyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
5-(morpholin-4-ylmethyl)-N-[2-(naphthalen-1-yl)ethyl]-1,2-oxazole-3-carboxamide
8-(propane-2-sulfonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(3-chlorophenyl)-4-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl}piperazine
7-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-3-methyl-3,4-dihydroquinazolin-4-one
N4,N4,5-trimethyl-N2-{[1-(prop-2-en-1-yl)pyrrolidin-3-yl]methyl}pyrimidine-2,4-diamine
7-fluoro-3-{[({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]methyl}-1,2-dihydroquinolin-2-one
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-[(1S,2S)-1,3-dihydroxy-1-phenylpropan-2-yl]urea
N-[3-(pyridin-3-yloxy)propyl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
1-(pyridin-2-ylmethyl)-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine
2-methoxy-N-(3-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}phenyl)acetamide
4-({[5-(4-fluorophenyl)-1,2,4-triazin-3-yl]amino}methyl)-1-(2-methoxyethyl)pyrrolidin-2-one
N-[3-(methylsulfanyl)phenyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
5-acetyl-N,2,4-trimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-pyrrole-3-carboxamide
2-[3-(cyclopropylmethyl)-5-(2,3-dimethyl-1H-indol-7-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
2-{2-[2-(4-fluorophenoxy)ethyl]phenoxy}-N-methylacetamide
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}acetamide
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(oxolan-2-ylmethoxy)ethan-1-one
1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-(3-phenylpyrrolidin-1-yl)ethan-1-one
9-(cyclopropylmethyl)-4-(4,6-dimethylpyridine-3-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(2-chlorophenyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-3-phenylpropanamide
4-methyl-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}-6H,7H,8H-cyclopenta[g]quinazoline
2-(4-{[cyclohexyl(methyl)amino]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(4-methoxypyrimidin-2-yl)pyrrolidin-3-yl]methanol
(3R,4R)-1-(3-methoxypyrazin-2-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-ol
N-{[5-(furan-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-methoxyacetamide
8-chloro-2-(furan-2-yl)-N-[(3-methyloxetan-3-yl)methyl]quinoline-4-carboxamide
[2-oxo-2-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)ethyl]urea