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5-[(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidine-3-carbonyl]-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
N-benzyl-2-methoxy-N-(1,3-thiazol-2-ylmethyl)pyridine-3-carboxamide
5-[1-(piperidin-1-yl)ethyl]-N-[2-(pyridin-2-yl)ethyl]furan-2-carboxamide
(1R,5R)-6-benzyl-3-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[1-(1H-pyrazol-1-yl)propan-2-yl]pyridin-2-amine
(2S)-N2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]pyrrolidine-1,2-dicarboxamide
4-(4-methylphenyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-(pyrimidin-5-yl)pyrimidin-2-amine
3-[(2S)-2-amino-3-methoxypropanamido]-N-ethyl-N-phenylbenzamide
1-(5-chloropyridin-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-[3-(3-chlorophenoxy)azetidine-1-carbonyl]-6-(2-methylpropyl)pyrimidin-2-amine
[1-(morpholin-4-yl)propan-2-yl]({[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl})amine
2-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)benzoic acid
N-(5-acetamido-2-fluorophenyl)-3-(morpholin-4-yl)azetidine-1-carboxamide
1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-3-(4-phenylazepane-1-carbonyl)-1,4-dihydropyridin-4-one
ethyl 4-[(4-methoxyphenyl)methyl]-1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidine-4-carboxylate
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-phenylacetamide
2-{4-[(1,7-dimethyl-1H-indol-3-yl)methyl]piperazin-1-yl}-5-methylpyrimidin-4-amine
1-ethyl-4-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-2-one
2-methyl-6-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
3-(5-{1-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1H-1,2,3-triazol-4-yl}thiophen-2-yl)prop-2-yn-1-ol
ethyl 5-{[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
2-amino-6-(3,4-dimethoxyphenyl)-4-[2-(methylsulfanyl)ethyl]pyridine-3-carbonitrile
N-[2-(5-methylfuran-2-yl)ethyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
3-methoxy-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-5-methoxypyridin-4-ol
2-(4-{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)pyrimidine
N-{[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
N-[3-(1H-indol-1-yl)propyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-[1'-(5-ethylthiophene-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
2-methoxy-1-{4-[2-(methylamino)benzoyl]-1,4-diazepan-1-yl}ethan-1-one
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
N-[1-(4-methoxyphenyl)propyl]-N,2-dimethylfuran-3-carboxamide
[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl){[5-(oxan-2-yl)furan-2-yl]methyl}amine
4-benzyl-3-ethyl-1-(1H-indole-5-carbonyl)-1,4-diazepan-5-one
(2S,4S)-1-benzyl-4-{[(2,5-dimethylphenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
1-(2-methanesulfonylethyl)-5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazole
({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)(1H-indol-2-ylmethyl)methylamine
N-[(5-methylfuran-2-yl)methyl]-3-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}propanamide
2,2-dimethyl-5-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]thiomorpholin-3-one
1-methyl-4-({4-methyl-5-[1-(piperidin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperazine
2-(4-{4-[(1,1-dioxo-1λ6-thiolan-3-yl)amino]piperidin-1-yl}phenyl)-N-[2-(2-methoxyphenyl)ethyl]acetamide
N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]quinoline-2-carboxamide
4-methyl-2-[2-(pyridin-3-yl)-1H-imidazol-1-yl]pyridine
6-amino-1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]hexan-1-one
methyl 2-(diethylsulfamoyl)-6-(2-ethylbutyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4,4,4-trifluoro-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
(1R,6S)-3-{3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzoyl}-9-methyl-3,9-diazabicyclo[4.2.1]nonane
1-benzyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
1-[(2S,4S)-1-[(2-methoxynaphthalen-1-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carbonyl]azepane