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(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(pyrrolidine-1-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
1-benzyl-4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-1,4-diazepan-6-ol
1-(cyclopropanesulfonyl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
1-[(4aR,8aS)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-decahydro-1,6-naphthyridin-6-yl]-4-phenylbutan-1-one
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylpropanamide
{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amine
1-cyclopentyl-4-[2-(thiophen-2-yl)pyrimidine-5-carbonyl]-1,4-diazepane
1-[(4-hydroxy-3-methoxyphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
7-(3,6-dimethylpyrazin-2-yl)-4-[(2S)-piperidine-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(2-methylphenyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1,4-diazepane-1-carboxamide
4-methyl-N-[(4-methylphenyl)(pyridin-4-yl)methyl]-1,2,5-oxadiazole-3-carboxamide
(cyclobutylmethyl)({[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
N4-[1-(thiophen-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine
4-cyclobutaneamido-N-methyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}benzamide
1-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[(3-propyl-1,2-oxazol-5-yl)methyl]urea
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-3-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-(morpholine-4-carbonyl)-N-(1,3-thiazol-2-ylmethyl)benzene-1-sulfonamide
1-methyl-4-({6-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]pyridin-3-yl}methyl)piperazine
N-{1-[1-(2-hydroxyacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-phenylmethanesulfonamide
2-[(5-methylpyrazin-2-yl)methyl]-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-benzyl-2-methyl-4-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-yl}pyrimidine
4-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)-1-cyclohexylpiperazin-2-one
2-(1-cyclohexyl-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
6-(2,5-dimethylbenzoyl)-N-[3-(2-oxoimidazolidin-1-yl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
5-ethyl-2-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}pyridine
methyl 3-[(2E)-3-(3-fluorophenyl)prop-2-enamido]-6-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
(1S,5R)-6-benzyl-3-(quinoxalin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2-(pyridin-2-yl)pyrimidine
2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
1-butyl-4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-2-one
3-[2-(3-fluorophenyl)ethyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,1,3,7-tetramethyl-1H-indole-2-carboxamide
(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-5-(9H-purin-6-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
6-methoxy-2,2-dimethyl-N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-4-amine
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethan-1-one
2-(2-phenylethyl)-8-(1H-pyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
3-benzyl-4-(5-chloro-2-fluorobenzoyl)piperazin-2-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}furan-3-carboxamide
4-(2-methoxyacetyl)-6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
3-(2-fluorophenyl)-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
4-(2-methylphenoxy)-1-[2-(pyridin-2-yl)acetyl]piperidine-4-carboxylic acid
N-[(3-ethoxy-4-methoxyphenyl)methyl]-N,1,4,6-tetramethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(4aS,8aR)-1-(piperidin-4-ylmethyl)-6-(trimethylpyrimidin-4-yl)-decahydro-1,6-naphthyridin-2-one
6-(1-methyl-1H-pyrazol-4-yl)-N2-(4-methylphenyl)-1,3,5-triazine-2,4-diamine
(4aR,6R,8aS)-8a-(methoxymethyl)-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-6-(morpholin-4-yl)-decahydroisoquinoline
1-[(4-chlorophenyl)methyl]-6-oxo-N-[3-(pyridin-4-yl)propyl]piperidine-3-carboxamide
1-[1-(2,2-dimethylpropyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
3-(2-methylphenyl)-1-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}piperidine
4-fluoro-3-{5-[(1S)-1-hydroxy-2-phenylethyl]-3-methyl-1H-1,2,4-triazol-1-yl}benzene-1-sulfonamide