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2-[(4-chlorophenyl)methyl]-8-(3-ethoxypropanoyl)-2,8-diazaspiro[4.5]decan-3-one
1-{[2-(4-chlorophenyl)-7-methoxyquinolin-3-yl]methyl}-1,4-diazepan-5-one
[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-(2-phenylethyl)piperidin-3-yl]methanol
1-[(2S)-2-(3-ethyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
4-({4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}methyl)-1,2-dihydrophthalazin-1-one
(2-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-oxoethyl)urea
1-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]-4-phenylbutan-1-one
(1S,6R)-N-[4-chloro-2-(trifluoromethyl)phenyl]-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
N-(3-hydroxy-3-phenylpropyl)-N,2-dimethylpyrimidine-5-carboxamide
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
2-[(4-chlorophenyl)sulfanyl]-1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
(3R,4S)-1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
ethyl 2-[2-(morpholine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]pyridine-3-carboxylate
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2-methylphenyl)methyl]piperidine
4-{1-[1-(2-ethyl-6-methylpyrimidin-4-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
1-(2-aminoethyl)-N-{2-[(4-chlorophenyl)methoxy]ethyl}-1H-1,2,3-triazole-4-carboxamide
2-(2-{1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
dimethyl(3-{3-[3-(pyridin-2-yl)phenyl]-1H-pyrazol-1-yl}propyl)amine
4-(8-methoxy-2H-chromen-3-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
[(3R,4R)-1-(3-fluoro-4-methoxybenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
(3S,4R)-1-[2-amino-6-(propan-2-yl)pyrimidine-4-carbonyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N,1,3-trimethyl-N-(2-phenyl-1-{1-[4-(thiophen-2-yl)butanoyl]piperidin-4-yl}ethyl)-1H-pyrazole-5-carboxamide
3-cyclohexyl-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1H-pyrazole-4-carboxamide
4-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-N-cyclopropylpiperazine-2-carboxamide
4-{[5-(1-cyclopentylpiperidin-3-yl)-1,2,4-oxadiazol-3-yl]methyl}morpholine
5-{1-[(3-ethoxy-2-hydroxyphenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
3-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridazine
methyl 2-{[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]amino}acetate
N-[2-(1-hydroxycyclopentyl)ethyl]-N-methyl-2-(1H-pyrrol-1-yl)propanamide
N-{2-[3-(ethylsulfanyl)-5-oxo-4,5-dihydro-1,2,4-triazin-6-yl]phenyl}-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
methyl 5-{[(1-carbamoylcycloheptyl)carbamoyl]amino}-2-chlorobenzoate
{[5-(methoxymethyl)furan-2-yl]methyl}(methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
ethyl 1-[(3-{[1-(thiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]piperidine-2-carboxylate
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-ethyl-N-[2-(phenylsulfanyl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-6-(2-fluorophenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
5-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-3-(4-methoxyphenyl)-1,2,4-oxadiazole
(1S,5R)-10-oxo-N-{3-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}-3,9-diazabicyclo[3.3.2]decane-3-carboxamide
2-fluoro-6-hydroxy-N-[1-(pyridin-4-yl)propyl]benzamide
(1S,5R)-3-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N3-[3-(dimethylamino)-2,2-dimethylpropyl]-1-(3-methylbutyl)-N5-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-ethyl-7-fluoro-N-(propan-2-yl)-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
1-ethyl-4-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1,2-dihydropyridin-2-one
N-(1-benzylpyrrolidin-3-yl)-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carboxamide
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-6-methoxyhexanamide
9-methoxy-7-(4-methylphenyl)-4-[(3-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-methoxy-N-{[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
N-methyl-N-(oxolan-2-ylmethyl)-2-(1H-1,2,4-triazol-1-yl)acetamide
3-{2-[3-(3-methylphenoxy)azetidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione