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3-(dimethyl-1,2-oxazol-4-yl)-1-{3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]morpholin-4-yl}propan-1-one
4-(1H-pyrazol-1-yl)-1-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}butan-1-one
3-(1-butyl-1H-imidazol-2-yl)-1-(4-chloro-2-fluorobenzoyl)piperidine
3-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-1-(pyridin-3-yl)urea
1-[3-(methylsulfanyl)propyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
[2-(dimethyl-1,3-thiazol-2-yl)ethyl]({[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-(pyrrolidin-3-yl)benzamide
1-(2,3-dimethylbenzoyl)-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
5-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
2-chloro-4-{1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
5-[5-(piperidin-1-ylmethyl)pyridin-2-yl]pyridin-2-amine
2-cyclohexyl-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-1,3-benzoxazole-6-carboxamide
1-ethyl-5-{[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl}-1H-1,2,4-triazole
N-(3-methyl-1-{7-propyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)pyridine-3-carboxamide
3-phenoxy-N-[1-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]propanamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(pyridin-4-yl)propanamide
1-(4-fluorophenyl)-N-(1,3-thiazol-2-ylmethyl)cyclopropane-1-carboxamide
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)piperidin-2-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
4-({5-[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
6'-carbamoyl-2'-oxo-7'-(pyrrolidin-1-yl)-2',3'-dihydro-1'H-spiro[cyclobutane-1,4'-quinoline]-3-carboxylic acid
1-[2-(1-butyl-1H-pyrazol-4-yl)quinoline-4-carbonyl]piperidine-4-carbonitrile
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-1-(4-hydroxy-4-phenylpiperidin-1-yl)ethan-1-one
(3aS,6aS)-2-(oxan-4-yl)-5-(pyrazin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(propan-2-yl)-5-[1-(2,3,4-trifluorophenyl)-1H-imidazol-2-yl]pyrimidin-2-amine
2-cyclohexyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1,3-benzoxazole-6-carboxamide
3-[5-(3-ethoxybenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-3-(2-oxopyrrolidin-1-yl)-N-(pyridin-4-ylmethyl)benzamide
5-methyl-1-[4-(5-methylpyrimidin-2-yl)phenyl]-1H-pyrazole-3-carboxylic acid
(1R,5S,8S)-N,N-dimethyl-3-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-3-azabicyclo[3.2.1]octan-8-amine
(2E)-3-(2-chlorophenyl)-N-[(3,4-dimethoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)prop-2-enamide
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}furan-2-carboxamide
(4aR,8aR)-2-(6-aminopyridine-3-carbonyl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
(3aR,6aR)-2-(cyclobutylmethyl)-5-(2,3-dimethylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(4-{[2-(pyridin-2-yl)ethyl]sulfanyl}phenyl)-1-[(1r,4r)-4-hydroxycyclohexyl]urea
N-[2-(1H-1,3-benzodiazole-1-carbonyl)phenyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
N-(1-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-2-phenylethyl)-N,2-dimethylfuran-3-carboxamide
3-methyl-8-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(cyclopropylmethyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
2-(1-tert-butyl-3-methyl-1H-1,2,4-triazol-5-yl)benzonitrile
8-methyl-N-[3-(1,3-oxazol-5-yl)phenyl]-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
(3S,4R)-4-methyl-1-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidine-3,4-diol
4-[4-(4-hydroxyphenyl)piperazine-1-carbonyl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
4-(1H-imidazol-2-ylmethyl)-2-(4-methylpentyl)morpholine
N-methyl-2-[4-(5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carbonyl)morpholin-3-yl]acetamide
1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}hex-5-yn-1-one
3-methoxy-1-{2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one