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N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
(1S,6R)-3-[(5-chloro-2,4-dimethoxyphenyl)methyl]-3,9-diazabicyclo[4.2.1]nonane
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-methyl-1H-pyrrole-3-carbonyl)piperidine
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(2S,4S)-4-amino-N-ethyl-1-[3-(1H-1,2,4-triazol-1-yl)adamantane-1-carbonyl]pyrrolidine-2-carboxamide
N-{1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]piperidin-4-yl}methanesulfonamide
benzyl({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}(methyl){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
4-(2,4-dioxoimidazolidin-1-yl)-N-[2-(5-methylfuran-2-yl)ethyl]benzamide
ethyl 5-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{1-[(2-chlorophenyl)methyl]-1H-pyrazol-5-yl}-3-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]urea
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
(3S,4R)-1-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
3-[1-(4-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]-6-methyl-1,2-dihydropyridin-2-one
3-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-6-methoxy-3,4-dihydroquinazolin-4-one
(2H-1,3-benzodioxol-4-ylmethyl)({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
3-(2H-1,3-benzodioxol-5-yl)-3-phenyl-N-[2-(pyrazin-2-yl)ethyl]propanamide
N-[4-(furan-2-yl)butan-2-yl]-N'-(4-methylphenyl)propanediamide
1-[2-(furan-2-yl)pyrrolidin-1-yl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
(3aS,6aR)-5-(4,6-dimethylpyrimidin-2-yl)-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
6-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
N4-[1-(4-chlorophenyl)ethyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
7-{[3-(butan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-4-methyl-3,4-dihydro-2H-1,4-benzoxazine
[(3R,4R)-4-[(dimethylamino)methyl]-1-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)pyrrolidin-3-yl]methanol
4-[2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carbonyl]-1,4-oxazepan-6-ol
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(9H-purin-6-yl)piperidin-4-amine
1-[(3-methylphenyl)methyl]-4-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]piperazine
2-(6-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyridin-3-yl)acetic acid
1-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-phenoxyethan-1-one
{2-[2-(2,6-dimethoxy-4-methylphenyl)phenoxy]ethyl}dimethylamine
(3S)-3-ethyl-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}morpholine
N-[2-(1,3-benzoxazol-2-ylsulfanyl)ethyl]-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
2-[benzyl({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidine
2-amino-6-(1-ethyl-1H-indol-3-yl)-4-(2-methyl-1H-imidazol-4-yl)pyridine-3-carbonitrile
1-(3,4-difluorobenzenesulfonyl)-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
3-(2-{2-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(4-methoxyphenyl)methyl]-4-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]morpholine
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-1-methyl-1H-indazole-3-carboxamide
2-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
(1R,5S,6R,7S)-N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
1-(2,3-dimethylphenyl)-4-{[4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}piperazine
1-[1-ethyl-5-(naphthalene-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
2-[2-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-3-ethyl-1,2-oxazole-5-carboxamide
N-(2-phenylethyl)-3-(thiophene-2-sulfonamidomethyl)piperidine-1-carboxamide
(1S,5R)-3-[(2E)-3-phenylprop-2-en-1-yl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-methoxyethyl)-1-methyl-5-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,3-benzodiazol-2-amine
2-(1,3-benzoxazol-2-yl)-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane