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1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decane
3-({[1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]oxy}methyl)pyridine
methyl[(4-methyl-1H-imidazol-2-yl)methyl]({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)amine
2-{6-[4-(1-ethoxyethyl)phenyl]pyridin-3-yl}acetic acid
4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1λ6-thiomorpholine-1,1-dione
{1-cyclohexyl-5-[3-(1H-imidazol-1-yl)propyl]-1H-1,2,4-triazol-3-yl}(phenyl)methanol
2-(morpholin-2-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}acetamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-ethyl-1H-pyrazole-5-carboxamide
5-methanesulfonyl-4-(piperidin-3-yl)-N-[3-(1H-pyrazol-1-yl)propyl]pyrimidin-2-amine
N-benzyl-4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
N-[1-(5-{[(4-methoxyphenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-3-methylthiophene-2-carboxamide
(4aS,7aR)-1-[2-(3-hydroxyphenyl)acetyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-(pyridin-2-ylmethyl)propanamide
4-(furan-2-yl)-2-[5-(methoxymethyl)-4-(3-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
1-ethyl-4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-3,5-dimethyl-1H-pyrazole
{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
1-{3-[5-(2-methylpropyl)-1H-1,2,4-triazol-3-yl]phenyl}ethan-1-one
N-[3-(2-ethylphenoxy)propyl]-N-methyl-2-(methylamino)pyrimidine-5-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2-(2-methoxyphenoxy)acetamide
(1R,5S)-6-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-6-azabicyclo[3.2.1]octane
3,4,4-trimethyl-1-{thieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-ol
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
2-(4-cycloheptanecarbonylmorpholin-3-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
N-[(2R,4R,6S)-2-cyclohexyl-6-[2-(2-hydroxyethoxy)phenyl]oxan-4-yl]acetamide
1-[(4-hydroxy-3,5-dimethylphenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
(3R,5S)-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
N-[2-({2-[(thiophen-2-ylmethyl)amino]phenyl}formamido)ethyl]acetamide
N-[2-(dimethylsulfamoyl)ethyl]-1-(4-methoxyphenyl)-2,2-dimethylcyclopropane-1-carboxamide
6-ethyl-N4-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-N2,N2-dimethylpyrimidine-2,4-diamine
2-(dimethylamino)-1-{4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}ethan-1-one
(3R,4R)-3-cyclobutyl-1-(1-cyclopropanecarbonylpiperidin-4-yl)-4-methylpyrrolidin-3-ol
1-[1'-(5-methyl-1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
3-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyridin-2-ol
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-(3-cyclopentylpropyl)propanamide
1-(cyclohexylmethyl)-3-hydroxy-3-{[(2-methylprop-2-en-1-yl)amino]methyl}piperidin-2-one
2-methyl-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-(morpholin-4-yl)propan-1-one
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(methylsulfamoyl)ethyl]pyrimidine-5-carboxamide
1-benzyl-N,N-dimethyl-5-[(1,3-thiazol-2-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(6-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridin-3-yl)ethan-1-one
4-({[3-(2-fluorophenyl)propyl]carbamoyl}amino)-N,N,3-trimethylbenzamide
N-(2-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}quinolin-5-yl)acetamide
2-ethyl-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3S,4S)-4-(morpholin-4-yl)-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-3-ol
2-{1-[(6-methylpyridin-2-yl)methyl]-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
2-(7-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]acetamide
4-(4-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
(2E)-N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enamide
3-(3-fluorophenyl)-N-(2-methoxyethyl)-N-[(2-methylphenyl)methyl]-1H-pyrazole-4-carboxamide
N-{[(2S,4S)-4-fluoro-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]pyrrolidin-2-yl]methyl}cyclobutanecarboxamide