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1-methyl-4-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
7-(3-chlorophenyl)-4-(2,2-dimethyloxane-4-carbonyl)-9-(thiophen-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[3-(3-methoxypropyl)piperidine-1-carbonyl]-5,7-dimethylquinolin-8-ol
5-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine
(3aS,6aS)-2-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-5-(2-methoxyacetyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[5-(4-chloro-2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-3-methoxypiperidine
4-methyl-6-(4-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}piperazin-1-yl)pyrimidin-2-amine
(2R,3R)-3-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-[1-(ethoxymethyl)-1H-pyrazol-4-yl]urea
N-cyclopentyl-2-{4-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]morpholin-3-yl}acetamide
N-ethyl-1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]pyrrolidine-3-carboxamide
7-{10,10-dichlorotricyclo[7.1.0.04,6]decane-5-carbonyl}-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
N-(4-methoxyphenyl)-3-{[(6-methylpyridin-2-yl)methyl]amino}-5-(methylsulfamoyl)benzamide
N-[4-({[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]acetamide
(1S,5R)-6-benzyl-3-[2-(2-methylphenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(6-methoxynaphthalen-2-yl)-4-methylmorpholine
ethyl 4-({3-[(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)oxy]phenyl}methyl)piperazine-1-carboxylate
1-(3-methoxypropyl)-8-[(4-methyl-1H-imidazol-2-yl)methyl]-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[7-(1-benzofuran-5-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methanamine
(3S,4S)-4-methoxy-1-[2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidin-3-ol
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]furan-2-carboxamide
14-(2-chloro-4-fluorophenyl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
(1R,7S)-3-[(3-methoxyphenyl)methyl]-6-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-[3-(4-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
N-{2-[(2-methyl-6-propylpyrimidin-4-yl)amino]ethyl}methanesulfonamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-3-yl]propanoic acid
8-[(2-chlorophenyl)methyl]-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
(2S,4S)-4-amino-N-methyl-1-{[1-phenyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(4-cyanophenyl)methyl]-4-propylpyrimidine-5-carboxamide
3-{1-[3-(dimethylamino)benzoyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
6-(4-{[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)pyridine-3-carbonitrile
3-{2-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-[4-(7-fluoro-2-methylquinoline-4-carbonyl)-1,4-diazepan-1-yl]-2-methoxyethan-1-one
2-{1-[(3,4-difluorophenyl)methyl]-4-[(5-ethylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N,N,1-trimethyl-6-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
2-methoxy-4-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]pyridine
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[3-(propan-2-yloxy)benzoyl]piperidin-3-yl]propan-1-ol
2-cyclobutanecarbonyl-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
2-(dimethylamino)-N-[(4,6-dimethylpyridin-2-yl)methyl]-2-(4-fluorophenyl)-N-methylacetamide
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
2-[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]-N-(2-methylphenyl)acetamide
N-cyclopentyl-1-{1-[6-(propan-2-yl)pyridazin-3-yl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
2-(1H-pyrrol-1-yl)-1-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]propan-1-one
3-(hydroxymethyl)-1-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}piperidin-3-ol
2-(4-methoxyphenyl)-5-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}pyrimidine
N-[2-(4-methylmorpholin-2-yl)ethyl]pentanamide
N-[(1S,2R)-2-(cyclooctylamino)cyclobutyl]-2-methyl-1,3-thiazole-4-carboxamide