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3-chloro-N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-4-fluoro-N-[(3S)-2-oxoazepan-3-yl]benzene-1-sulfonamide
(3aR,7aS)-5-methyl-2-[4-(1H-pyrazol-1-yl)benzenesulfonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-{1'-[(2E)-3-phenylprop-2-en-1-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
2-[4-(3-chloropyridin-2-yl)-1-[(2-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl][(2,3,5-trimethyl-1H-indol-7-yl)methyl]amine
1-[5-methoxy-2-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
1-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(pyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
3-[4-(2-methylphenoxy)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
5-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-(2-methoxy-5-{[3-(pyridin-2-yl)azetidin-1-yl]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
4-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-2-one
N-[(2S,4R,6S)-2-[2-(methylamino)pyridin-3-yl]-6-(2-phenylethyl)oxan-4-yl]acetamide
1-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-4-yl)-2-phenylethan-1-ol
1-[(4-methoxypyridin-2-yl)methyl]-3-[4-(3-methylpiperidine-1-carbonyl)phenyl]urea
4-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-1-(4-methylphenyl)piperazin-2-one
5-(1H-imidazol-1-ylmethyl)-2-[2-(piperidin-1-ylmethyl)phenoxy]pyridine
1-(2,5-dimethylfuran-3-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
N-[1-(3-methylphenyl)piperidin-4-yl]-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
1-(diethylamino)-3-[2-methoxy-4-({[2-(3-methoxyphenyl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-(2-methanesulfonamidoethyl)-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
N-(2,6-dimethoxypyridin-3-yl)-3-[(2-methylphenyl)methoxy]azetidine-1-carboxamide
N-[(4-fluorophenyl)methyl]-5-[1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]thiophene-2-carboxamide
4-chloro-3-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(1R,5R)-6-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-phenyl-1,2-oxazole-5-carboxamide
2-(4-{1-[2-(1H-pyrrol-1-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)ethan-1-ol
7-[(8-chloro-4-hydroxyquinolin-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
7-[2-(1H-imidazol-2-yl)benzoyl]-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-(1-methylpiperidin-2-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
8-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
4-({3-[2-(dimethylamino)ethyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)-1-ethyl-1H-pyrrole-2-carbonitrile
3-[1-(4-amino-5-methylpyrimidin-2-yl)piperidin-4-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-benzyl-3-{1-[(2-ethylpyrimidin-5-yl)methyl]piperidin-4-yl}-N-methylpropanamide
2-methyl-6-{1-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidin-4-yl}pyrimidin-4-ol
4-(2-{[1-(4-fluorophenyl)cyclopropyl]formamido}ethyl)benzoic acid
8-chloro-N,2-dimethyl-N-[1-(pyridin-3-yl)propyl]quinoline-4-carboxamide
7-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
methyl 3-(4-methoxybenzamido)-5-{[(3-methoxyphenyl)methyl]amino}-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-({4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-N,N-dimethyl-1,3-thiazol-2-amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
5-(4-chlorophenyl)-3-(pyrrolidin-1-yl)-1,2,4-triazine
2-{5-[2-(3-chloro-1H-1,2,4-triazol-5-yl)ethyl]-1-(3-fluorophenyl)-1H-1,2,4-triazol-3-yl}acetamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
1-{2-oxo-2-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethyl}-1,2-dihydropyrimidin-2-one
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-2-(1H-1,2,4-triazol-1-yl)benzamide
3-{5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}phenol