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2-(thiomorpholin-4-yl)-2-(2,3,4-trimethoxyphenyl)acetic acid
N-[4-(2-fluorophenoxy)phenyl]-1-[(3-hydroxyphenyl)methyl]piperidine-4-carboxamide
2-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-4-methylphenol
2-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1H-imidazole
2-(2,4-dioxo-1,3-thiazolidin-3-yl)-N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
9-(5,6-dimethylpyrimidin-4-yl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[2-(1H-pyrazol-1-yl)ethyl]-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine
4-{2-[1-(4-fluorophenyl)-1H-1,2,4-triazol-5-yl]ethyl}pyridine
2-(2,3-dimethylphenyl)-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]acetic acid
3-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-4-(2-methylpyrrolidine-1-carbonyl)quinoline
2-[3-({3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
2-(2-phenylethyl)-8-[2-(propan-2-yloxy)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
[3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)-2,4,6-trimethylphenyl]methanol
2-benzyl-8-(1-methyl-1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)-N-ethylcyclopropanamine
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(pyrrolidine-1-sulfonyl)-decahydro-1,6-naphthyridin-2-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}acetamide
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]acetamide
1-[(1R,5R)-6-[3-(benzyloxy)propyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(8aS)-2-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})amine
N-[(4-hydroxyphenyl)methyl]-2-methyl-N-(pyridin-4-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
N-[3-(2-cyclopropyl-1H-imidazol-1-yl)phenyl]-2-phenylacetamide
5-{[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]sulfonyl}-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
[(3R,4R)-1-[4-(dimethylamino)naphthalene-1-carbonyl]-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-[(2-chlorophenyl)methyl]-1-cyclopropyl-6-oxopiperidine-3-carboxamide
6-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyrazine-2-carboxamide
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decane
4-(4-fluorophenyl)-1-[(5-propylfuran-2-yl)methyl]piperidin-4-ol
4-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
N-(1-benzothiophen-2-ylmethyl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
(4aS,7aR)-1-(4-chloro-2-fluorobenzoyl)-4-(cyclopropylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(cyclohex-1-en-1-ylmethyl)acetamide
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
2-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}-6-methoxyphenol
4-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
ethyl 4-[(2-chlorophenyl)methyl]-1-(2-hydroxyethyl)piperidine-4-carboxylate
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(furan-2-carbonyl)pyrrolidin-3-yl]methanol
2-(dimethylamino)-2-(2-fluorophenyl)-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}acetamide
1-[2-(4-chlorophenyl)ethyl]-N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-6-oxopiperidine-3-carboxamide
6-(2-methylquinolin-5-yl)pyridin-2-amine
N-methyl-3-{[(oxan-4-yl)amino]methyl}-N-[2-(pyridin-2-yl)ethyl]pyridin-2-amine
N3-(2,1,3-benzothiadiazol-5-ylmethyl)-N1,N1-dimethylpiperidine-1,3-dicarboxamide
1-[1-(furan-3-ylmethyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine