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2-[(1-hydroxycyclohexyl)methyl]-4-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
(2R)-2-amino-N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}propanamide
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
(1R,5S,8R)-3-(3-phenylpropyl)-3-azabicyclo[3.2.1]octan-8-ol
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-[3-(pyridin-3-yl)phenyl]propanamide
2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]pyrimidin-4-amine
N-(1-{7-[3-(1,3-benzothiazol-2-yl)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
5-(4-methoxyphenyl)-3-(4-propylpiperazin-1-yl)-1,2,4-triazine
(3R,4S)-1-[(4-methoxypiperidin-1-yl)sulfonyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
6-methyl-3-(3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-1,2-dihydropyridin-2-one
(2S)-2-(methoxymethyl)-N-(2-phenyl-1,3-benzoxazol-5-yl)pyrrolidine-1-carboxamide
2-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{5-[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]-3-methyl-1H-1,2,4-triazol-1-yl}pyridine
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]oxolane-2-carboxamide
1,3-dimethyl-5-[({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)methyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-(2H-1,3-benzodioxol-5-yl)-1-[(4-ethynylphenyl)methyl]piperidin-3-amine
methyl 8-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
dimethyl({[4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-1,4-oxazepan-6-yl]methyl})amine
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(morpholin-4-yl)butan-1-one
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
2-(dimethylamino)-N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2-methyl-1-[4-({2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}amino)piperidin-1-yl]propan-1-one
N-{4-[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]phenyl}ethane-1-sulfonamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
(3aS,6aS)-2-[(3-chloro-4-methoxyphenyl)methyl]-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-ethyl-4-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)piperazine
N-(propan-2-yl)-3-{5-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-{[1-butyl-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]methyl}piperidin-3-ol
1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
4-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-6-(propan-2-yl)pyrimidine
(3R,4R)-4-(azepan-1-yl)-1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-3-ol
3-ethyl-5-{[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-4,5-dihydro-1,2-oxazole
1-(2-methoxyacetyl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-3-carboxamide
2-[2-({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amino)ethyl]-6-phenyl-2,3,4,5-tetrahydropyridazin-3-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-[4-(methylsulfanyl)phenyl]acetamide
(2R,3R,6R)-5-(isoquinolin-5-ylmethyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(3-chloro-1,2-oxazol-5-yl)-1-[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]propan-1-one
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-methylpiperidine-3-carboxamide
3,5-dimethyl-2-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-1H-indole
N-{4-[4-(dimethylamino)phenyl]-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl}acetamide
1-[(1-{6-[ethyl(methyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-[3-(morpholin-4-yl)propyl]-5-(1,2-oxazinane-2-carbonyl)piperidin-2-one
3-(1-ethyl-1H-pyrazol-3-yl)-4-(4-methoxy-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R,4S)-1-(3-fluoro-4-methoxybenzenesulfonyl)-3,4-dimethylpiperidin-4-ol
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-2,3-dimethyl-N-(pyridin-4-ylmethyl)-1H-indole-7-carboxamide
5-[(2-phenyl-1,3-oxazol-4-yl)methyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-chloro-N-(2-methoxyethyl)-4-({1-[1-(5-methylpyridin-2-yl)propan-2-yl]piperidin-4-yl}oxy)benzamide
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one