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4-{3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}quinoline
2-methyl-2-(4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}phenyl)propanenitrile
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]but-2-ynamide
1-[7-(1-benzothiophen-3-yl)-9-(pyridin-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-[(5-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]-3,3-dimethylurea
3,4-dimethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
4-({[6-(methoxymethyl)pyrimidin-4-yl]amino}methyl)benzene-1-sulfonamide
N,6-dimethyl-2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
1-(2-{[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]amino}ethyl)piperidine-3-carboxamide
2-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-5-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinoline
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-4-(pyridin-4-yl)pyrimidin-2-amine
(3aS,6aS)-2-[(1-ethyl-1H-indol-5-yl)methyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
(4-{[4-phenyl-5-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}phenyl)methanol
2-(2,5-dioxoimidazolidin-1-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}acetamide
5-{2-[(3-chlorophenyl)methyl]pyrimidin-4-yl}-2-ethoxybenzoic acid
4-methyl-2-[1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidin-4-yl]-1H-1,3-benzodiazole
3-(2-methoxyacetamido)-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)benzamide
3-{[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}quinoline
3-(1-methanesulfonylpiperidin-4-yl)-1-(2-phenylphenyl)urea
3-methyl-N-[(3-methylthiophen-2-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
N-cyclopropyl-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-(2-{imidazo[1,2-a]pyrimidin-2-yl}ethyl)propanamide
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-8-azabicyclo[3.2.1]octane
3-phenyl-4-[2-(propan-2-yl)-1,3-oxazol-4-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
methyl({[4-(pyridin-3-yl)phenyl]methyl}){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
3-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
2-{3-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]phenoxy}acetamide
3-{[1-(furan-3-ylmethyl)piperidin-4-yl]methyl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl[(2-methylpyridin-4-yl)methyl]{[5-(oxolan-2-yl)thiophen-2-yl]methyl}amine
2-methyl-9-(2-phenoxyethanesulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[(2-methoxyethyl)sulfamoyl]-5-(pyridin-4-yl)benzoic acid
7-(cyclobutylmethyl)-2-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-(3-fluorophenyl)-4-[3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]pyrrolidin-2-one
1-{[(3-phenylprop-2-yn-1-yl)(propyl)carbamoyl]methyl}piperidine-4-carboxamide
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-4-(1H-indol-2-ylmethyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
N-[(1-benzylpiperidin-3-yl)methyl]-6-(morpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-(2H-1,2,3-benzotriazol-2-yl)-1-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]ethan-1-one
7-[(2-fluorophenyl)methyl]-2-[(2-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
5-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-1H-1,3-benzodiazole
N-methyl-1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]-N-(thiophen-3-ylmethyl)piperidine-4-carboxamide
3-{methyl[1-(3-methylpyridin-2-yl)propan-2-yl]amino}-N-(pyridin-3-yl)propanamide
{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}(thiophen-3-ylmethyl)amine
N-[2-(dimethylsulfamoyl)ethyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-3-[(3-methylbutyl)amino]-5-(phenylsulfamoyl)benzamide
5-ethyl-2,3-dimethyl-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine
[(3,4-dimethoxyphenyl)methyl](methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
4-(hydroxymethyl)-1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-ol