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N-[2-(N-methylmethanesulfonamido)ethyl]-2,3-dihydro-1-benzofuran-5-carboxamide
2-(benzyloxy)-N-(1,4-dioxan-2-ylmethyl)acetamide
(4S)-3,3,4-trimethyl-1-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}piperidin-4-ol
2-(2-fluoro-6-methoxyphenyl)pyridine-4-carboxamide
2-(1H-imidazol-1-yl)-1-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}ethan-1-one
2-(5-methoxyfuran-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-[4-(3,6-dimethylpyrazin-2-yl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
3-methyl-1-(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2-dihydroquinoxalin-2-one
[2-(1-methyl-1H-pyrazol-4-yl)ethyl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
N-(1,2-oxazol-3-ylmethyl)-3-{[2-(pyrrolidin-1-yl)ethyl]sulfamoyl}benzamide
4-{2-[(1-cyclopentylpiperidin-3-yl)formamido]ethyl}benzoic acid
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(methylsulfanyl)benzamide
3-(N-methylmethanesulfonamido)-N-[1-(3-methylpyridin-2-yl)ethyl]propanamide
N-(furan-2-ylmethyl)-N-methyl-1-[2-(2-methyl-1,3-benzothiazol-5-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
8-(dimethyl-1,2-oxazole-4-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-cyclopropyl-4-{[3-(1-methyl-1H-pyrazol-4-yl)propyl]sulfamoyl}benzamide
N-[2-(pyridin-3-yloxy)ethyl]-2,3-dihydro-1-benzofuran-5-carboxamide
1-ethyl-N-{3-[methyl(phenyl)amino]propyl}piperidine-2-carboxamide
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-4-(trifluoromethyl)pyrimidin-2-amine
2-{6-[(dimethylamino)methyl]-1,4-oxazepane-4-carbonyl}-5-fluorophenol
5-[ethyl(2-methylprop-2-en-1-yl)amino]-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-(3-chlorophenyl)-9-hydroxy-N,N-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-sulfonamide
4-(1-hydroxypropan-2-yl)-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
4-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
(3S,4R)-N,N-dimethyl-1-{[3-(methylsulfanyl)phenyl]methyl}-4-propylpyrrolidin-3-amine
1-(1-benzofuran-2-ylmethyl)-4-phenoxypiperidine-4-carboxylic acid
3-[(4,4-difluoropiperidin-1-yl)methyl]-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-{4-[(4-chlorophenyl)methyl]-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl}acetic acid
8-(butan-2-yl)-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2,3-dihydro-1H-inden-2-yl)-5-[2-(ethylamino)ethyl]pyrrolidin-2-one
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-4-(1H-pyrazol-4-yl)butanamide
1-(2-hydroxyethyl)-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1H-1,3-benzodiazole-5-carboxamide
N-{[3-(2-methoxyethyl)-1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-N-(4-methylphenyl)methanesulfonamide
N-{[1-(oxan-4-yl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide
3-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-N-phenylpropanamide
N-cyclopropyl-2-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]pyridine-4-carboxamide
methyl (2S)-1-{5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}pyrrolidine-2-carboxylate
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
4-(1,3-benzothiazol-2-ylmethyl)-2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-6-chloroimidazo[1,2-a]pyridine-2-carboxamide
1-[(3S,7S)-3-(hydroxymethyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-trien-5-yl]-4-phenylbutane-1,4-dione
2-fluoro-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-5-sulfamoylbenzamide
{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}amine
N-(2-methylphenyl)-3-(1,8-naphthyridin-2-ylformamido)propanamide
N-{2-[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}acetamide
1-({1-[6-(2,5-dihydro-1H-pyrrol-1-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
3-methyl-4-(naphthalen-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(4-methoxy-2-methylphenyl)-3-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(3-methoxyphenyl)-N-methyl-N-(thian-4-yl)-1H-pyrazole-5-carboxamide
[2-(2,3-dimethylphenoxy)ethyl][(4-methanesulfonylmorpholin-2-yl)methyl]amine