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(3S,4S)-1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
11-[(1-methyl-1H-pyrazol-4-yl)methyl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-12-one
(1R,2R)-2-[3-(2-ethoxyethyl)-5-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-1,2,4-triazol-1-yl]cyclohexan-1-ol
N,N,4-trimethyl-3-({[1-(2-methylpropyl)cyclopropyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-benzyl-4-cyano-N-(1,1-dioxo-1λ6-thiolan-3-yl)-1H-pyrrole-2-carboxamide
4-(1-hydroxypropyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-(2-methylpropyl)acetamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,3-dimethyl-1H-pyrazole-4-carboxamide
3-(2-phenoxyethyl)-8-{spiro[2.3]hexane-1-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S)-1-ethyl-3-methyl-4-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)piperazin-2-one
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
N-(2-hydroxyethyl)-3-(1-methylpiperidin-2-yl)-N-(1,3-thiazol-2-ylmethyl)propanamide
3-[(1H-1,3-benzodiazol-2-ylmethyl)(ethyl)amino]-1λ6-thiolane-1,1-dione
1-[(2E)-2-methylbut-2-en-1-yl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
{4-[3-(1-methoxyethyl)phenyl]pyridin-2-yl}methanol
3-{4-[(5-chlorofuran-2-yl)methyl]piperazin-1-yl}-1λ6-thiolane-1,1-dione
4-{3-[2-(3,5-difluoro-4-methoxyphenyl)-1H-imidazol-1-yl]phenyl}-4H-1,2,4-triazole
[(4-methoxy-2,5-dimethylphenyl)methyl]({3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl})amine
1-(2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
2-({[1-(4-chloro-2-fluorobenzoyl)piperidin-3-yl]oxy}methyl)pyridine
4-[(2-fluorophenyl)methyl]-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1,4-diazepan-5-one
3-{2-[2-(morpholin-4-ylmethyl)piperidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]-N-[1-(naphthalen-1-yl)ethyl]propanamide
4-[4-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)piperazin-1-yl]quinazoline
(5S,9aS,9bS)-5-(4-hydroxyquinolin-2-yl)-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
{3-[(3-methoxyphenyl)methyl]-1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl}methanol
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](methyl){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[1-(dimethylamino)-2-methylpropan-2-yl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[(2-methylphenyl)sulfanyl]-N-(4H-1,2,4-triazol-4-yl)acetamide
3-hexyl-8-(pyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-1-[(3R)-piperidin-3-yl]urea
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-3-amine
5-(2,4-difluoro-3-methoxyphenyl)-1-propyl-1H,4H-pyrazolo[3,4-d]imidazole
ethyl 4-[(4-chlorophenyl)methyl]-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylate
(3aR,6aR)-2-cyclopentyl-5-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(3-fluorophenyl)methyl]-4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperazin-2-one
4-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole
5-(3-propylmorpholine-4-carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[(1R,2R)-2-(benzyloxy)cyclopentyl]-1-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
N1-{1-[4-(3-fluorophenyl)phenyl]piperidin-4-yl}propane-1,3-diamine
7-[(2-fluorophenyl)methyl]-2-(6-methylpyridine-3-carbonyl)-2,7-diazaspiro[4.5]decane
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(2-hydroxypropanoyl)piperidine-4-carboxamide
1-[(4aR,8aS)-1-(5-methyl-1H-indole-2-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-2-methoxyethan-1-one
4-methoxy-2-(4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperazin-1-yl)pyrimidine
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[(1S)-2-hydroxy-1-phenylethyl]-1,2-oxazole-3-carboxamide
1-(2-methylpropyl)-5-oxo-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyrrolidine-3-carboxamide
1-methyl-2-[1-(pyridin-2-ylmethyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
2-[3-(oxolan-3-yl)-5-[(2-oxopiperidin-1-yl)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[(3-methylphenyl)methyl]amino}methyl)piperidin-2-one
3-{[1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]formamido}propanamide