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ethyl 3-[(2,4-difluorophenyl)methyl]-1-[2-(1H-pyrazol-1-yl)acetyl]piperidine-3-carboxylate
(2R)-2-amino-N-cyclopropyl-4-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pentanamide
N-[(2-methylphenyl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-[2-(3-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-N-[2-(morpholin-4-yl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
[1-(1H-1,3-benzodiazole-5-carbonyl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-[(3R,4S)-1-[2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)(quinolin-5-ylmethyl)amine
ethyl 4-benzyl-1-(pyridin-4-ylmethyl)piperidine-4-carboxylate
5-(4-phenyl-1-{[1-(prop-2-en-1-yl)pyrrolidin-3-yl]methyl}-1H-imidazol-5-yl)-2-propylpyrimidine
1-ethyl-5-{1-[1-(1,3-thiazol-2-yl)ethyl]-1H-imidazol-2-yl}-1H-1,2,4-triazole
N,2-dimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
4-(2-{4-[3-(thiophene-2-carbonyl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)morpholine
N-{5-[1-(methoxymethyl)cyclobutaneamido]-2-methylphenyl}-4-methylbenzamide
3-{1-azabicyclo[3.2.1]octan-5-yloxy}benzonitrile
2-{3-[3-(3-methylpyridin-4-yl)phenyl]-1H-pyrazol-1-yl}ethan-1-ol
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(1,2,4-oxadiazol-3-yl)piperidine
[(3S,5R)-5-[(dimethylamino)methyl]-1-[(6-methylquinolin-5-yl)methyl]piperidin-3-yl]methanol
(1S,5R)-3-[2-(3-chloro-4-fluorophenoxy)acetyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S)-N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-2-amino-3-(1H-indol-3-yl)propanamide
1-[3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-benzyl-5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-N-ethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(6-methoxypyridin-3-yl)acetic acid
1-(1-cyclopropanecarbonylpiperidine-4-carbonyl)-2-(3-fluorophenyl)azepane
5-(1H-indol-1-ylmethyl)-N-methyl-N-[2-(oxan-2-yl)ethyl]-1H-pyrazole-3-carboxamide
4-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-amine
methyl 2-[4-(2-methylphenoxy)piperidine-1-carbonyl]piperidine-1-carboxylate
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N-methyl-2-(1H-pyrazol-1-yl)butanamide
(3S,4R)-1-[(5-ethylfuran-2-yl)methyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-methoxyquinoline-4-carboxamide
ethyl 1-[2-(methylsulfanyl)acetyl]-3-(3-phenylpropyl)piperidine-3-carboxylate
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
N-(cyclopropylmethyl)-1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-methylpiperidine-3-carboxamide
1-(furan-2-ylmethyl)-4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperazine
N-{[1-(oxan-4-yl)piperidin-4-yl]methyl}-2,3-dihydro-1-benzofuran-7-carboxamide
1-cyclopropyl-4-{4-[(4-ethoxyphenyl)methyl]piperazine-1-carbonyl}pyrrolidin-2-one
2,5-dimethyl-N-[1-(4-methylpyridin-2-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-methyl-4-phenyl-9-[2-(pyrrolidin-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
(4aS,7aR)-1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[1'-(2-methyl-5-propylpyrimidin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
4-{[4-(4-fluorophenyl)-1,4-diazepan-1-yl]methyl}phenol
N-tert-butyl-2-[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]benzene-1-sulfonamide
(1S,5R)-6-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(4aS,8aR)-1-(2-aminoethyl)-6-(1-benzofuran-5-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
5-{3-[1-(pyridin-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine