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2-methyl-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)-1,3-thiazole-4-carboxamide
4-methoxy-N-[(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)methyl]benzene-1-sulfonamide
4-hydroxy-N-methyl-2-(phenoxymethyl)-N-(thiophen-3-ylmethyl)pyrimidine-5-carboxamide
4-[(1-methoxybutan-2-yl)amino]-N-(2-methoxyethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-(2-methylpyridine-3-carbonyl)-4-(2-methylquinolin-6-yl)piperidin-4-ol
5-methyl-1'-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}-N-[2-(2-oxoimidazolidin-1-yl)ethyl]benzamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]-1H-pyrazole-3-carboxamide
3-[1-(4-methoxyphenyl)-3-methyl-1H-pyrazol-5-yl]-1-[1-(4-methyl-1H-imidazol-2-yl)propyl]urea
3-cyclohexyl-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-[(5-chloro-2,4-dimethoxyphenyl)methyl]-N-methyloxan-4-amine
(3S,4R)-1-[2-chloro-5-(trifluoromethyl)benzoyl]-N,N-dimethyl-4-propylpyrrolidin-3-amine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylfuran-2-carboxamide
1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-(3-fluorobenzoyl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
(1S,5R)-6-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(4-fluorophenyl)-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidin-3-amine
2-(1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethan-1-ol
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)-2-(pyrrolidin-1-yl)benzamide
(1S,5R)-6-(cyclopropylmethyl)-3-[(4-methoxy-2,5-dimethylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aS,7aR)-1-(3-aminopropanoyl)-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(azocan-1-yl)-3-[2-methoxy-4-({[2-(3-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
1'-(5-ethylthiophene-2-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 4-{[4-(quinazolin-4-yl)piperazin-1-yl]methyl}thiophene-2-carboxylate
1-(4-fluorophenyl)-6,6-dimethyl-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
6-[1-(2-benzyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]pyrimidin-4-ol
2-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-N-(5-methylpyridin-2-yl)acetamide
6-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]pyridine-2-carbonitrile
5-(2-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}phenyl)-1H-1,2,3,4-tetrazole
2-ethyl-6-methyl-1-[(5-methylfuran-2-yl)methyl]-3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-7-acetamido-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
N-(1-methyl-1H-indazol-5-yl)-3-(1,2,3,6-tetrahydropyridin-1-ylmethyl)benzamide
2,5-dimethyl-4-(3-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
N-(propan-2-yl)-6-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
4-methyl-9-[2-(pyridin-3-yl)acetyl]-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
2-amino-1-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpropan-1-one
5-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyrazin-2-ol
(1S,5R)-6-(cyclobutylmethyl)-3-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(3-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-oxopropyl)pyrrolidin-2-one
(1S,5R)-3-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(2,3-dihydro-1H-inden-4-yl)-1-[1-(furan-2-carbonyl)piperidin-4-yl]urea
N'1-methyl-N'1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}cyclopropane-1,1-dicarboxamide
2-methyl-5-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methoxy}-1,3-benzothiazole
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(1H-1,2,4-triazol-1-yl)acetamide
1-{3-[4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-3-oxopropyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
6-methyl-5-{1-[(1-methylpyrrolidin-3-yl)methyl]-1H-imidazol-2-yl}quinoline
5-acetamido-2-ethyl-N-(oxolan-3-yl)-1-(pyridin-3-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-5-(morpholin-4-ylmethyl)furan-3-carboxamide
4-[(5-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazol-3-yl)methyl]morpholine
3-(5-aminopentyl)-7-methyl-3H,4H-thieno[3,2-d]pyrimidin-4-one