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{1-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-N-(oxolan-3-yl)-1H-pyrazole-4-carboxamide
4,5-dimethyl 1-[(3S,5S)-1-[(3-ethoxy-4-methoxyphenyl)methyl]-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
8-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]benzamide
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-4-(pyrrolidin-1-ylmethyl)benzamide
N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
N-(2-methoxyethyl)-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
6-methyl-2-({1-oxo-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-2-yl}methyl)-4H-pyrido[1,2-a]pyrimidin-4-one
7-(cyclopropylmethyl)-2-[4-(furan-2-yl)benzoyl]-2,7-diazaspiro[4.5]decane
[(3-chlorophenyl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(oxolan-2-ylmethyl)amine
1-(2,5-dimethylfuran-3-carbonyl)-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-ethoxy-4-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}phenol
N-cyclopropyl-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
1-methyl-3-propyl-N-{[4-(trifluoromethoxy)phenyl]methyl}-1H-pyrazole-5-carboxamide
N-methyl-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-N-(thiophen-3-ylmethyl)piperidine-4-carboxamide
2-[(1S,5R)-6-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
3-{[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]sulfonyl}benzonitrile
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}pyridine
2-{5-[(1R)-1-aminoethyl]-3-(4-chlorophenoxymethyl)-1H-1,2,4-triazol-1-yl}acetic acid
N-{[2-(2-benzamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
1-(cyclohexylmethyl)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-6-oxopiperidine-3-carboxamide
1-{[4-(methylsulfanyl)phenyl]methyl}-3-(1H-pyrazol-5-yl)piperidine
3-fluoro-4-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
2-(1-methyl-4-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-yl)pyridine
[(3S,5R)-1-(2,3-dihydro-1H-indene-5-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-2-[4-methyl-3-(5-methylthiophen-2-yl)-1H-pyrazol-1-yl]acetamide
5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[1-(pyridin-4-ylmethyl)piperidin-4-yl]pyridin-2-amine
4-[(2-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}phenyl)methyl]morpholine
1-{2-[(3-chlorophenyl)methyl]-1,3-benzoxazole-6-carbonyl}-N,N-diethylpyrrolidin-3-amine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-(furan-2-yl)-N-methyl-2-oxoacetamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-(1-propylpiperidin-4-yl)acetamide
3-ethyl-2-[2-(trifluoromethyl)morpholine-4-carbonyl]-1H-indole
(furan-2-ylmethyl)[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](thiophen-3-ylmethyl)amine
2-(4-methyl-6-{[2-(pyrrolidine-1-sulfonyl)ethyl]amino}pyrimidin-2-yl)phenol
(1-methoxypropan-2-yl)({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl})amine
3-(pyridin-4-yl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
3-[1-(5-chlorothiophene-2-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
4-[2-(morpholin-3-yl)acetyl]-1-(2-phenylphenyl)piperazin-2-one
5-[(2-methylphenyl)methyl]-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
N-(2-ethoxybutyl)-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-[(2-fluorophenyl)methyl]-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,4-diazepane
7-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-methyl-1H-pyrazolo[1,5-a]imidazole
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-[(1-methyl-1H-indol-2-yl)methyl]pyrrolidin-3-amine
2-(3-methoxyphenoxymethyl)-4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1,3-oxazole
2-(4-fluorophenyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
1-(2-methylpropyl)-5-(3-phenylbutanoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
5-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-2-(propan-2-yl)-1,3-benzoxazole