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4-[(1,2-oxazol-3-ylmethyl)sulfamoyl]-N-[(3S)-piperidin-3-yl]benzamide
4-{3-[(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)oxy]benzoyl}morpholine
4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-2-amine
1-[3-(benzyloxy)azetidin-1-yl]-2-(1-ethylpiperidin-4-yl)ethan-1-one
2-methyl-N-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}imidazo[1,2-a]pyridine-6-carboxamide
5-[1-(2,5-dimethoxyphenyl)-1H-imidazol-2-yl]-2-(pyrrolidin-1-yl)pyrimidine
4-(hydroxymethyl)-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidin-4-ol
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(dimethyl-1,2-oxazol-4-yl)acetamide
3-[(3R,4S)-4-(morpholin-4-yl)-1-(5-propylthiophene-3-carbonyl)piperidin-3-yl]propanoic acid
9-ethyl-4-[5-(methoxymethyl)furan-2-carbonyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(3aR,5S,6S,7aS)-2-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)-octahydro-1H-isoindole-5,6-diol
1-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-[2-(pyridin-2-yl)ethyl]piperazine
2-(2,3-dihydro-1H-inden-1-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}acetamide
2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5-(trifluoromethyl)pyridine
9-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2,3-dimethyl-1H-indole-7-carboxamide
3-[2-(2,4-difluorophenyl)ethyl]-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine
N-(2-{7-[(3,5-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-(4-fluorophenyl)acetamide
(3S,4R)-3-benzyl-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-methylpiperidin-4-ol
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-(piperidin-3-yl)benzamide
N2,N2-diethyl-6-(pyridin-4-yl)pyrimidine-2,4-diamine
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(2-methoxybenzoyl)piperidine-3-carboxylate
N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
5-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-(1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-1-oxopropan-2-yl)pyrrolidin-2-one
(3S,4S)-1-(4-methoxybenzoyl)-4-{methyl[2-(oxan-4-yl)ethyl]amino}pyrrolidin-3-ol
(3R,5R)-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
N,N-dimethyl-4-{1-[3-(1H-pyrazol-5-yl)phenyl]piperidin-4-yl}piperazine-1-carboxamide
2-(4-{1-[(4-methoxyphenyl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)pyridine
4-{1-[(4-phenyl-1,3-thiazol-2-yl)methyl]azetidin-3-yl}morpholine
(4aS,8aR)-6-(6-methylpyridazin-3-yl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
2-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]benzonitrile
2-[(4-methoxypiperidin-1-yl)sulfonyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-1,4-diazepane
1-methyl-1'-[1-(propan-2-yl)piperidine-3-carbonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-(1-ethylpiperidin-4-yl)-1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
2-[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-4,6-dimethylpyridine-3-carboxylic acid
5-acetyl-N-[3-(cyclohexylsulfanyl)propyl]thiophene-3-carboxamide
4-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)pyrimidine
N-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
1-{5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
N-(1H-1,3-benzodiazol-2-ylmethyl)-3-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-N-methyl-1,2-oxazole-5-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-[2-(pyridin-4-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-(propylamino)pyridine-3-carboxamide
methyl 5-[(1-methoxypropan-2-yl)amino]-3-(oxolane-2-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-{[benzyl(methyl)amino]methyl}-N-(1,4-dioxan-2-ylmethyl)-N-methyl-1,2-oxazole-3-carboxamide
1-{[4-(methylsulfanyl)phenyl]methyl}-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
1-[(3,5-dimethylphenyl)methyl]-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperazin-2-one
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)piperidin-2-one
2-{[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-methyl-1H-1,3-benzodiazole