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(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(2,3-difluorophenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-phenyl-1-[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]piperazine
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(2-methylbutan-2-yl)acetamide
4-methyl-2-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
1-{[4-(2-methylphenyl)phenyl]methyl}-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
N-(3,4-dimethylphenyl)-2-{[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)amino}acetamide
4,5,6-trimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(methylsulfanyl)ethan-1-one
4-(1H-imidazol-1-yl)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidine-4-carboxylic acid
N-cyclohexyl-4-[2-(pyridin-3-yl)-1H-imidazol-1-yl]benzamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(1-methyl-1H-imidazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-(but-2-ynoyl)-N-phenyl-6-azaspiro[2.5]octane-1-carboxamide
N-{2-[1-(2-fluorophenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
2-(3-chlorophenoxy)-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-[7-(1,3-benzothiazol-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxyethan-1-one
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N-methylbenzamide
3-{1-[(3,4-dimethylphenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
5-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-2-methyl-1,4-dihydropyridin-4-one
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]quinoline-2-carboxamide
3-[1-(3-cyclopentylpropyl)piperidin-4-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[2-({[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
(2R,6S)-2,6-dimethyl-4-(1-{5-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidin-4-yl)morpholine
N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-2-(ethylamino)pyrimidine-5-carboxamide
2-({2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}methyl)-8-fluoroquinolin-4-ol
(1R,5R)-6-propyl-3-(5-propyl-1,3,4-thiadiazol-2-yl)-3,6-diazabicyclo[3.2.2]nonane
(2S)-4-methyl-2-({6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazol-3-yl}formamido)pentanamide
(1R,5R)-N,N-dimethyl-6-(trimethyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-4-(oxan-4-yl)piperazine
(1R,5R)-3-(1,2-oxazole-3-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(thiophen-3-yl)ethan-1-one
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]amine
N-[(7-{[4-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-5-(methoxymethyl)furan-2-carboxamide
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(diphenylmethyl)-1H-1,2,3-triazole-4-carboxamide
1'-(3-methoxy-4-methylbenzoyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-3-(2-methoxyphenyl)propanamide
N3-(butan-2-yl)-1-cyclopentyl-4-oxo-N5-[2-(propan-2-yloxy)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
4-cyclopentyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]pyrimidin-2-amine
4-[2-(4-amino-3,5-dimethyl-1H-pyrazol-1-yl)ethoxy]-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
3-(azocan-1-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}propanamide
4-(hydroxymethyl)-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}pyridine-2-carboxamide
[(5-chloro-3-methyl-1H-indol-2-yl)methyl](methyl)[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
2-(2,3-dimethylphenoxy)-N-[2-(N-methylmethanesulfonamido)ethyl]acetamide
N-methyl-N-({3-methyl-1-[2-(4-methylpiperazin-1-yl)ethyl]-1H-pyrazol-4-yl}methyl)-2,3-dihydro-1H-inden-2-amine
2-{4-[3-(cyclopropylcarbamoyl)piperidin-1-yl]piperidin-1-yl}pyridine-3-carboxamide
N-[(2-fluorophenyl)methyl]-3-(1-methanesulfonylpiperidin-3-yl)propanamide
1-cyclopentyl-4-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-2-one
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)piperidin-2-one
1-(4-{4-[3-(1H-imidazol-1-yl)pyrrolidin-1-yl]piperidin-1-yl}phenyl)-5-methylpyrrolidin-2-one
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[(2-chloro-6-fluorophenyl)methyl]piperidine