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{4-[(4-chlorophenyl)methyl]-1-(2-phenylethyl)piperidin-4-yl}methanol
4-(3,4-dimethoxyphenyl)-3-(1H-indol-3-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(1H-pyrazol-1-yl)propan-2-yl]-2-(pyridin-4-yl)quinoline-4-carboxamide
1-ethyl-5-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
6-{methyl[(3-methylthiophen-2-yl)methyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-2-(2-oxo-1,2-dihydroquinolin-1-yl)acetamide
8-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-1-oxa-8-azaspiro[4.5]decan-3-ol
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(propan-2-yl)acetamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
6-methyl-2-[2-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-3,4-dihydropyrimidin-4-one
N,N-dimethyl-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrazin-2-amine
(1-{1-[4-(3-fluorophenyl)phenyl]piperidin-4-yl}piperidin-3-yl)methanol
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}thiophene-3-carboxamide
2-[(3-methoxyphenyl)methyl]-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]morpholine
3-[(3R,4S)-4-(dimethylamino)-1-[4-(2-methoxyphenyl)benzoyl]piperidin-3-yl]propan-1-ol
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl){[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
methyl 3-(7-chloro-2-{[2-(1H-1,2,4-triazol-1-yl)acetamido]methyl}-2,3-dihydro-1-benzofuran-5-yl)benzoate
1-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,4-dimethyl-1H-indole
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[2-(3-methyl-1H-1,2,4-triazol-5-yl)acetyl]pyrrolidine-3-carboxylic acid
(2R)-2-cyclohexyl-1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-hydroxyethan-1-one
2-(3-methoxypyridin-2-yl)benzonitrile
1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-3-(4-methyl-1,4-diazepan-1-yl)propan-1-one
4-[4-(azocane-1-carbonyl)piperidin-1-yl]-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
methyl 3-({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)propanoate
4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-6-[(3-fluorophenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
ethyl 1-ethyl-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
5-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
2-cyclobutyl-1-{6-hydroxy-4-[(4-methyl-1H-imidazol-2-yl)methyl]-1,4-diazepan-1-yl}ethan-1-one
7-(2-methoxyethyl)-2-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-1-[4-(thiophen-2-ylmethoxy)phenyl]urea
2-(1-{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)ethan-1-ol
(5-fluoro-7-{pyrazolo[1,5-a]pyrimidin-3-yl}-2,3-dihydro-1-benzofuran-2-yl)methanamine
4-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
N-(furan-2-ylmethyl)-5-{[2-(2-methoxyphenyl)ethyl]amino}-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N,N-dimethyl-7-(2-methylbenzoyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
5-ethyl-2-({4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)pyridine
{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(2-phenoxyethyl)piperidin-3-yl}methanol
ethyl 4-[(2-chlorophenyl)methyl]-1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}piperidine-4-carboxylate
2-(4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
3-(3-fluoro-4-methoxybenzoyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
1-(3-{4-[(3-hydroxyphenyl)methyl]piperazine-1-carbonyl}piperidin-1-yl)-2-methoxyethan-1-one
7-(3-methoxypropyl)-2-(6-methylpyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(azepan-1-yl)-3-[3-({[(2-methoxyphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
1-(3-chlorophenyl)-5-[2-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,4-triazole
3-methyl-N-{1-[1-(1H-pyrazol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
methyl 5-(2-methoxy-4-methylbenzenesulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
[(2S,4R)-1-[(3-chloropyridin-4-yl)methyl]-4-(dimethylamino)pyrrolidin-2-yl]methanol
1-methyl-9-(2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one