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1-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)-3-methylpiperidine-3-carbonitrile
1-[9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2,2-diphenylethan-1-one
6-methyl-5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-2-oxo-1,2-dihydropyridine-3-carbonitrile
1-methyl-4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazol-5-amine
N-(2,3-dihydro-1H-inden-2-yl)-4-(propylsulfamoyl)benzamide
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
4-[2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-benzofuran-5-yl]-1-(thiophen-3-ylmethyl)piperidin-4-ol
(2R)-2-amino-1-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
1-methyl-3-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-6-yl}-1-[1-(pyridin-3-yl)pentyl]urea
2-methyl-5-(3-{[4-phenyl-5-(propan-2-yl)-1H-imidazol-1-yl]methyl}pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
3-{[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]methyl}benzoic acid
1-{2-oxo-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-4-phenylpyrrolidin-2-one
3-{2-[4-(4-fluorophenyl)-4-hydroxypiperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-(cyclopropylmethyl)-6-methyl-2-(4-methylphenoxymethyl)-1-[2-(morpholin-4-yl)ethyl]-4-oxo-N-propyl-1,4-dihydropyridine-3-carboxamide
3-(1H-indazol-1-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
4-(1H-1,2,3,4-tetrazol-1-ylmethyl)-N-(2,2,2-trifluoroethyl)benzamide
3-cyclopentyl-1-(3-{3-oxo-3-[4-(pyridin-2-yl)piperazin-1-yl]propyl}piperidin-1-yl)propan-1-one
3-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonane-7-carbonyl]-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
1-(prop-2-en-1-yl)-5-({5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-(cyclohex-1-en-1-yl)-1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-{[(2-methylprop-2-en-1-yl)amino]methyl}piperidin-2-one
N-[2-(1-methylpiperidin-3-yl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
1-(5-{3-[2-(3-fluorophenyl)ethyl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
1-ethyl-6-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}-1H-indole
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[(1-methyl-1H-indol-5-yl)methyl]pyrrolidin-3-yl]methanol
5-acetyl-3-[2-(4-fluorophenyl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amine
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1H-pyrazol-4-yl)propanamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]acetamide
4-{2-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-1λ6-thiane-1,1-dione
2-amino-4-{2-[3-(dimethylamino)propoxy]phenyl}-6-(propan-2-yl)pyridine-3-carbonitrile
(1R,2S,6R,7S)-4-(1,3,4-thiadiazol-2-yl)-4-azatricyclo[5.2.2.02,6]undecane
3-(1H-1,3-benzodiazol-2-yl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylpropanamide
4-methyl-1-{2-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydroquinolin-2-one
3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}-1-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]propan-1-one
N-cyclopentyl-2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carboxamide
2-cyclohexyl-5-[1-(1H-imidazol-2-ylmethyl)-1H-1,2,3-triazol-4-yl]pyrimidine
2-(2-methyl-1,3-thiazol-4-yl)-N-{3-[4-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenoxy]propyl}acetamide
(2S,4R)-1-[(2,4-difluorophenyl)methyl]-N-[2-(dimethylamino)ethyl]-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
methyl 2-{2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}acetate
N-ethyl-1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-3-carboxamide
2-({4-[(benzyloxy)methyl]-1H-1,2,3-triazol-1-yl}methyl)morpholine
N-butyl-N-methyl-3-({methyl[3-(morpholin-4-yl)propyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
2-(4-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}morpholin-2-yl)ethan-1-amine
1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(diethylamino)propan-1-one
N-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-propyl-1H-pyrazole-4-carboxamide
2-benzyl-8-methanesulfonyl-2,8-diazaspiro[5.5]undecan-3-one
N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-4-(4H-1,2,4-triazol-3-yl)piperidine