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N-({2-[(dimethylamino)methyl]phenyl}methyl)-5-ethyl-N-methyl-1,3,4-oxadiazol-2-amine
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)(3-methylbut-2-en-1-yl)amine
1-[2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-3-ol
[2-(1H-imidazol-1-yl)ethyl](methyl){[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}amine
N-{2-[(1-cyclohexylpiperidin-3-yl)formamido]ethyl}pyridine-3-carboxamide
N3-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1-cyclopentyl-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-(2-methyl-1H-imidazol-1-yl)-1-{2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}butan-1-one
N-[1-(2,5-difluorophenyl)cyclopropyl]-4-hydroxy-1-methylpiperidine-4-carboxamide
2-methoxy-3-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidin-3-ol
4-({5-[2-(methylsulfanyl)propyl]-4-phenyl-1H-imidazol-1-yl}methyl)-1H-indole
2-{1-ethyl-2,4-dioxo-8-[(3-phenoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-8-[(3-methylphenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-(2-phenylethyl)-2-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-2,7-diazaspiro[4.5]decane
N-(6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-(2-{[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}ethyl)imidazolidin-2-one
(3aR,6aR)-2-(cyclobutylmethyl)-5-(6-cyclopropylpyrimidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(pyrrolidine-1-carbonyl)piperidine-4-carboxylic acid
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpropanamide
(1R,5S)-6-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-6-azabicyclo[3.2.1]octane
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)spiro[2.4]heptane-1-carboxamide
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-7-methylquinolin-2-ol
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-(quinolin-2-ylmethyl)benzamide
N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-(thiophen-2-yl)propanamide
N-methyl-N-(2-phenoxyethyl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-(4-methoxypiperidin-1-yl)pyridine
1-(6-methyl-2-propylpyrimidin-4-yl)-1,4-diazepan-5-one
N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
4-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)piperazine-2-carboxylic acid
1-cyclopentanecarbonyl-N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-amine
N-{[1-(3-cyanopyridin-2-yl)piperidin-3-yl]methyl}-3,5-dimethoxybenzamide
N-[2-(2,6-dimethylphenoxy)ethyl]-N-methyl-3-(1-methylpiperidin-2-yl)propanamide
3-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-1H-indole
1-{6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridin-3-yl}ethan-1-one
4-(3,4-difluorobenzenesulfonyl)-9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1R,5S,8S)-N-(2-chloro-5-sulfamoylphenyl)-8-methoxy-3-azabicyclo[3.2.1]octane-3-carboxamide
3-butyl-4-(5-methoxyfuran-2-carbonyl)-1-methylpiperazin-2-one
N-[(3R,4R)-4-hydroxypiperidin-3-yl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
1-[4-(pyridin-2-yl)piperazin-1-yl]-3-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-3-yl]propan-1-one
(1S,5R)-6-benzyl-3-(5-methyl-1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
6-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}pyridine-3-carbonitrile
4-(4-{[2-(1H-pyrazol-1-yl)ethyl]amino}piperidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
3-(2H-1,3-benzodioxol-5-yl)-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]propan-1-one
[(5-phenyl-1,2-oxazol-3-yl)methyl]({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
3-acetamido-N-methyl-N-[(3-methylthiophen-2-yl)methyl]benzamide
3-amino-1-[(3-chloro-4-ethoxyphenyl)methyl]pyrrolidine-3-carboxylic acid
4-{5-methyl-2-oxo-4-[2-(pyridin-4-ylsulfanyl)acetyl]piperazin-1-yl}benzonitrile
8-(1,3-benzothiazol-2-ylmethyl)-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4S)-4-amino-1-[3-(3,4-dimethylphenyl)propanoyl]-N-ethylpyrrolidine-2-carboxamide
2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-N,N-bis(prop-2-en-1-yl)acetamide