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1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-(3-phenylpropyl)-1,4-diazepane
2-[(1-hydroxypropan-2-yl)amino]-N-(2-methoxy-5-methylphenyl)acetamide
1-ethyl-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2,3-dihydro-1,4-benzodioxine-2-carboxamide
1-(azepan-1-yl)-3-{4-[({imidazo[1,2-a]pyridin-3-ylmethyl}amino)methyl]-2-methoxyphenoxy}propan-2-ol
4-(1-benzofuran-2-ylmethyl)-N-(cyclohexylmethyl)morpholine-2-carboxamide
1-benzyl-4-[1-(4-methylphenyl)cyclopropanecarbonyl]-1,4-diazepan-6-ol
4-{[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]methyl}benzoic acid
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one
6-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine-2,4-diamine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(methylsulfanyl)pyrimidin-4-amine
2-({2-[(2H-1,3-benzodioxol-5-ylmethyl)(cyclopentyl)carbamoyl]phenyl}amino)acetic acid
2,7,8-trimethyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}quinoline-4-carboxamide
2-(1-cyclopentyl-4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperazin-2-yl)ethan-1-ol
5-acetyl-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}thiophene-3-carboxamide
N-methyl-1-(3-phenylpropyl)-N-[(2,4,5-trimethoxyphenyl)methyl]piperidin-3-amine
1-[2-(dimethylamino)-6-(pyrrolidin-3-ylmethyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
N-[2-(7-{[5-(hydroxymethyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-4-methoxybenzamide
4-methoxy-3-(1,2,3,4-tetrahydroisoquinolin-5-yl)benzoic acid
ethyl 4-[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]piperidine-1-carboxylate
ethyl 5-(2-acetamidoacetyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[1'-(4-chloro-3-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-(4-hydroxy-4-phenylpiperidin-1-yl)-3-(1-methylpiperidin-2-yl)propan-1-one
5-(naphthalen-1-yl)-3-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]-1,2,4-triazine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(1R,2R)-2-hydroxycyclohexyl]propanamide
4-methyl-N-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-5-{1-[2-(thiophen-2-yl)ethyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]({4-[2-(3-methylpiperidin-1-yl)ethoxy]phenyl}methyl)amine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl})amine
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-(2-hydroxyphenoxy)acetamide
3-methoxy-N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]propanamide
5,6,7-trimethoxy-4-[(1s,4s)-4-aminocyclohexyl]-1,2,3,4-tetrahydroquinolin-2-one
1-[2-(dimethylamino)acetyl]-4-(3-methylbutyl)-1,4-diazepane-6-carboxylic acid
2-(5-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
N-{2-methyl-1-oxo-1-[4-(pyridin-3-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-2-yl}thiophene-2-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-(2-methylpropyl)benzamide
1-[3-(2-methoxyphenyl)propyl]-3-[4-(2-oxopyrrolidin-1-yl)phenyl]urea
4-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}piperazin-2-one
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}thian-4-amine
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-(3-methyl-1H-1,2,4-triazol-5-yl)ethan-1-one
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-2-methoxyacetamide
N-[1-(4-{[(3-methoxyphenyl)methyl](methyl)carbamoyl}phenyl)-1H-pyrazol-4-yl]oxolane-3-carboxamide
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}({2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl})amine
1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}-2-(4-methylpiperidin-1-yl)ethan-1-one
2-(2,5-dimethylphenoxy)-N-methyl-N-[4-(morpholin-4-yl)butyl]propanamide
8-{[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]methyl}-3-oxatricyclo[7.3.1.05,13]trideca-1(12),5(13),6,8,10-pentaen-2-one
N-benzyl-N-(cyclopropylmethyl)-1-(diphenylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-benzyl-8-(furan-3-ylmethyl)-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)pyrazolo[1,5-a]pyridine-3-carboxamide
1-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-(2-methylpropyl)pyrrolidin-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide