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3-({2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}methyl)-N-(1-ethyl-1H-pyrazol-5-yl)benzamide
1-[(3-methylphenyl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(3-methylphenyl)methyl]piperazin-2-one
N-[(3S,4R)-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide
2-(3,4-dichlorophenyl)-4-(1H-pyrrole-2-carbonyl)morpholine
methyl 3-{6-[(3-methoxyphenyl)methoxy]-2-oxo-4-[3-(prop-2-en-1-yloxy)benzoyl]-1,4-diazepan-1-yl}propanoate
1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
1-({3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}carbonyl)cyclopropane-1-carboxamide
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-3-methyl-5,6-dihydro-1,4-dioxine-2-carboxamide
2-(dimethylamino)-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-(4-methylphenyl)acetamide
2-[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
4-(1-methyl-1H-pyrrole-2-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 5-[1-(pyridine-4-carbonyl)piperidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-(4-fluoro-2-methylbenzoyl)-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
7-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-2-oxa-7-azaspiro[4.5]decan-8-one
4-{4-[(3,4-dimethoxyphenyl)methyl]piperazin-1-yl}-2-[1-(thiophen-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-(4-fluorobenzenesulfonyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
1-{1-[(3-fluoro-5-methylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
N-({1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-[4-(oxolan-2-yl)butyl]urea
N-{[1-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
1-(4-{[2-(1H-imidazol-1-yl)ethyl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
3-methyl-8-{2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(thiophen-2-ylmethyl)piperidine
N-cyclopentyl-4,6-dimethyl-2-oxo-N-(3-phenylprop-2-yn-1-yl)-1,2-dihydropyridine-3-carboxamide
ethyl 1-(5-acetylthiophene-3-carbonyl)-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylate
1-(3-{[(2,1,3-benzothiadiazol-5-ylmethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-1-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-phenyl-1H-imidazole
1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
(2R,6R)-4-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-{1-[3-(1H-indol-1-yl)propyl]-1H-1,2,3-triazol-4-yl}phenol
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-4-(pyridin-4-yl)pyrimidin-2-amine
4-(3-{1-oxa-8-azaspiro[4.5]decan-8-yl}-3-oxopropyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
5-(methoxymethyl)-N-[(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]furan-2-carboxamide
[1-(2-fluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methanol
3-(5-{[(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amino]methyl}thiophen-3-yl)prop-2-yn-1-ol
4-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-3-methoxyphenol
N-(2,2-diphenylpropyl)-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide
methyl 3-({[1-(4-chlorophenyl)cyclobutyl]formamido}methyl)-5-(pyrazine-2-amido)benzoate
2-(5-methyl-1-propyl-1H-pyrazol-4-yl)-6-(1-methylpiperidin-3-yl)-3,4-dihydropyrimidin-4-one
2-amino-6-cyclopropanecarbonyl-4-[5-(hydroxymethyl)furan-2-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
methyl 3-[(3,3-dimethylbutanamido)methyl]-5-phenylmethanesulfonamidobenzoate
(4aS,8aR)-6-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
ethyl 3-{[1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propanoate
N-cyclopentyl-3-{5-[(2S)-2,3-dihydroxypropyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-(4-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
5-{2-[(2-phenoxyethyl)amino]ethyl}-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-one
1-(5,6-dimethylpyrimidin-4-yl)-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol