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N-cyclopropyl-2-[(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)oxy]-4-methoxybenzamide
1-[4-(4-chlorophenoxy)piperidin-1-yl]-3-(1H-imidazol-1-yl)butan-1-one
2-amino-1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-methylpropan-1-one
N-cyclohexyl-3-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)propanamide
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{5-[2-(1,1-dioxo-1λ6-thiolan-3-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-(2-methoxyethyl)-N-methyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
3-[1-(4-chlorobenzoyl)piperidin-4-yl]-N-[(4-fluorophenyl)methyl]propanamide
3-{1-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
2-[4-(6-methyl-2-propylpyrimidin-4-yl)-1H-pyrazol-1-yl]-N-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}acetamide
3-(4-methoxy-2-methylbenzoyl)-1-(propane-2-sulfonyl)piperidine
2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-1,3-benzodiazole
(1R,2R,6S,7S)-4-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
13-(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)-4,6-dimethyl-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-11-one
2-(2,3-dihydro-1H-indol-1-yl)-2-oxo-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}acetamide
1-(4-{[(2-methylphenyl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)oxolane-2-carboxamide
1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyridin-3-ylmethyl)piperazine
1-(carbamoylmethyl)-N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]piperidine-3-carboxamide
2-(dimethylamino)-N,N-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-sulfonamide
3-{2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-oxoethyl}-2,6,6-trimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indol-4-one
1-[4-(2-ethoxyphenyl)piperazin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
8-{[4-(2-hydroxyethoxy)phenyl]methyl}-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)morpholin-3-yl]-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]acetamide
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}amine
4-(2-methyl-1H-imidazol-1-yl)-1-(9H-purin-6-yl)piperidine-4-carboxylic acid
N-({1-[(2,4-dimethylphenyl)methyl]piperidin-4-yl}methyl)-2,2-dimethylpropanamide
N-{[7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-(morpholin-4-yl)cyclohexane-1-carboxamide
2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
methyl (2S,4S)-4-(2-fluorobenzamido)-1-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidine-2-carboxylate
(4aS,7aR)-1-(2-hydroxyacetyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3-propyl-1,2-oxazol-5-yl)methyl]-6-(thiomorpholin-4-yl)pyridine-3-carboxamide
1,5-dimethyl-4-{[methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}-1H-pyrrole-2-carbonitrile
2-{2-[3-(hydroxymethyl)-3-methylpiperidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
N-methyl-N-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,4-tetrahydronaphthalen-1-amine
(2S,4R)-4-(3-hydroxybenzamido)-1-(1H-imidazol-4-ylmethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-ethyl-8-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-chloro-2-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
1-[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
1-[1-(4-cyanophenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
1-(4-{2-[(2-methylphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)pentane-1,4-dione
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-(2-methylphenoxy)ethan-1-one
1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-(morpholin-3-yl)ethan-1-one
3-chloro-4-hydroxy-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}benzamide
4-{1-[3-(3-methoxyphenyl)phenyl]piperidin-4-yl}piperazin-2-one
2,2-diphenyl-1-[4-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]ethan-1-ol
4-{5-[1-(piperidin-1-yl)ethyl]furan-2-carbonyl}thiomorpholine
({5-[(4-chlorophenyl)sulfanyl]furan-2-yl}methyl)({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl})amine
2-[3-(4-methanesulfonylphenyl)-4-methoxyphenyl]ethan-1-amine