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N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
2-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-4,6-dimethylpyridine-3-carbonitrile
2,5-dichloro-N-{2-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}benzamide
{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl})amine
1-[(2-fluorophenyl)methyl]-6-oxo-N-[4-(pyridin-2-yl)butyl]piperidine-3-carboxamide
6,7-dimethoxy-2-[1-(2-methylpropyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
3-[2-(dimethylamino)ethyl]-8-(2,2-dimethylpropyl)-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[2-(1-ethyl-1H-pyrazol-4-yl)quinoline-4-carbonyl]-1,3-dimethylpiperazin-2-one
1-[4-(4-methylphenoxy)piperidin-1-yl]-3-(1-methylpiperidin-3-yl)propan-1-one
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-[1-(4-methylphenyl)piperidin-4-yl]-decahydro-2,7-naphthyridine-2-carboxamide
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-3-(1-methylpiperidin-2-yl)propanamide
4-methoxy-N-(2-methoxyethyl)-2-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
1-(furan-2-carbonyl)-4-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-1,4-diazepane
2-methyl-8-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecane
3-cyano-N-{[(3S,4S)-3-hydroxy-1-(3-methylfuran-2-carbonyl)piperidin-4-yl]methyl}benzamide
3-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}thiomorpholine
N-cycloheptyl-5-(4-fluorophenyl)-1,2,4-triazin-3-amine
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(oxan-4-yl)ethyl]acetamide
4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(furan-2-ylmethyl)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}piperidine-3-carboxamide
3-methoxy-1-[2-(3-phenylpyrrolidin-1-yl)ethyl]piperidine
(1-benzothiophen-2-ylmethyl)({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
N-[(1-hydroxycyclohexyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
(2S,4S)-4-amino-N,N-diethyl-1-[2-hydroxy-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]pyrrolidine-2-carboxamide
1-(6-aminopyrimidin-4-yl)-4-[(2-methoxyethyl)carbamoyl]-1,4-diazepane-6-carboxylic acid
N-{[2-(4-acetylpiperazin-1-yl)-7-methylquinolin-3-yl]methyl}-N-cyclopropyl-2-(trifluoromethyl)benzamide
(2S,4S)-N,N-diethyl-1-methyl-4-[4-(pyrrolidin-1-yl)benzamido]pyrrolidine-2-carboxamide
N-[1-(3-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-oxoethyl}-2-azaspiro[4.4]nonan-3-one
4-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
[(3R,5R)-5-(morpholin-4-ylmethyl)-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidin-3-yl]methanol
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(2-methoxypyrimidin-5-yl)methyl]-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-(2,6-dimethylpyridin-3-yl)-2-[3-(1H-imidazol-2-yl)piperidin-1-yl]pyrimidine
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-2-methyl-1,3-thiazole-4-carboxamide
4-{[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N-methyl-1,3-thiazol-2-amine
6-{[(1-ethylpyrrolidin-2-yl)methyl]amino}-N-methyl-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
(1S,5R)-3-[(6-ethoxyquinolin-2-yl)methyl]-3,9-diazabicyclo[3.3.2]decan-10-one
4-methoxy-N-(2-methoxyethyl)-2-[(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)oxy]benzamide
4-[2-(3-fluoro-4-phenylphenyl)propanoyl]-3-(2-hydroxyethyl)piperazin-2-one
3-hydroxy-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-1-(3-phenylpropyl)piperidin-2-one
3-(2-hydroxyphenyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-pyrazole-5-carboxamide
3-(3,4-dimethyl-1H-pyrazol-5-yl)-N-[(5-methylfuran-2-yl)methyl]propanamide
3-acetamido-N-[2-(2-phenoxyethoxy)phenyl]propanamide
N-[(3S,4R)-1-(5-chloropyridine-2-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
7-(1-benzothiophen-3-yl)-4-(2-hydroxyethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-ethyl-N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-methyl-1,3-thiazole-5-carboxamide
3-(5-methylfuran-2-yl)-1-[(3-methylphenyl)methyl]-5-(pyrrolidin-3-yl)-1H-1,2,4-triazole