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N-[(3-methoxyphenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{[1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}-1,2-dihydropyridin-2-one
4-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]-1-(furan-2-ylmethyl)piperidine
N-({4-[(4-methoxyphenyl)methyl]-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl}methyl)-N-methylmethanesulfonamide
2-(4-methoxy-3-methylphenyl)-6-(piperidine-1-carbonyl)pyrazine
(3S)-4-(3,5-difluoropyridine-2-carbonyl)-3-ethylmorpholine
4-{1-[6-(4-fluorophenyl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
2-methyl-4-[3-(3-phenylpiperazine-1-carbonyl)phenyl]butan-2-ol
(4aS,8aR)-6-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
5-benzyl-5-{3-[4-(hydroxydiphenylmethyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
5-(3-methoxyphenyl)-N-[2-phenyl-2-(piperidin-1-yl)ethyl]-1,2,4-triazin-3-amine
5-(2,6-difluorophenoxymethyl)-N-[2-(2,4-dimethoxyphenyl)ethyl]-1,2-oxazole-3-carboxamide
3-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2-dimethyl-1H-indol-5-ol
methyl (2S,4R)-4-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-amido]-1-methylpyrrolidine-2-carboxylate
2-(2-{[4-(thiophene-2-carbonyl)piperazin-1-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
2-({[3-(4-fluorophenyl)oxolan-3-yl]methyl}amino)-N-(pyrazin-2-yl)acetamide
7-[2-(2,3-dihydro-1H-indol-1-yl)-2-oxoethyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
2-(dimethylamino)-7-(2-hydroxypropanoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
diethyl({2-ethyl-5-[4-(1,3,5-triazin-2-yl)piperazine-1-carbonyl]furan-3-yl}methyl)amine
5-methoxy-1-methyl-2-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1H-indole
2-oxo-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-phenyl-1,2-dihydropyridine-3-carboxamide
[2-(1H-imidazol-1-yl)ethyl](methyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}piperidine
N-cyclopentyl-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)cyclobutanecarboxamide
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-3-({2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)benzamide
1-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-2-[4-(4-fluorophenyl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]ethan-1-one
2,5-dimethyl-3-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}pyrazine
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,2,3-benzotriazole-5-carboxamide
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[3-(1H-1,2,4-triazol-1-yl)propyl]pyrimidine-5-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-[1-(furan-2-ylmethyl)piperidin-4-yl]-3,6-diazabicyclo[3.2.2]nonane
3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-2-ethoxypyridine
N-(1H-imidazol-2-ylmethyl)-N,4-dimethyl-5-phenylthiophene-2-carboxamide
2-{5-[6-amino-2-(morpholin-4-yl)pyrimidin-4-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
[2-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-1,3-thiazol-4-yl]methanol
N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-2-methyl-N-(pyridin-4-ylmethyl)-1,3-benzoxazole-6-carboxamide
4-chloro-N-{2-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}benzene-1-sulfonamide
1-(3-methylbutyl)-8-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-cyclopropanecarbonyl-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]piperidine-4-carboxamide
N6-cyclopentyl-N5-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-{[(1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
8-[(1S,3R)-3-aminocyclopentanecarbonyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine-4-carboxamide
N-{[2-(4-acetylpiperazin-1-yl)-7-methylquinolin-3-yl]methyl}-N-cyclopropyloxolane-2-carboxamide
N-(1-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
[1-(3,5-difluorophenyl)ethyl][2-(4-methoxyphenoxy)ethyl]amine
2-cyano-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}benzamide
2-[(2S)-2-hydroxypropanoyl]-N-[(5-methylfuran-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide