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3-{1-[(2-chlorophenyl)methyl]-1H-pyrazol-5-yl}-1-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]urea
N-(2,2-diphenylethyl)-1-ethyl-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-(cyclohexylmethyl)-2-[3-(methylsulfanyl)propyl]-2,7-diazaspiro[4.5]decan-6-one
2-[1-(5-chloropyridine-2-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
1-{[4-(2,2-dimethylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
(1s,4s)-4-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]cyclohexan-1-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(5-ethylpyridin-2-yl)methyl]piperidin-3-ol
2-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-octahydropyrrolo[1,2-a]piperazine
4-{1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-yl}piperazin-2-one
1-cyclopentyl-N-[3-(4H-1,2,4-triazol-4-yl)propyl]piperidine-3-carboxamide
2-(5-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
N-(4-methoxyphenyl)piperidin-3-amine
2-amino-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-methylpropanamide
(4aS,7aR)-1-[2-(1H-pyrazol-1-yl)acetyl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-chloro-6-methylphenyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
5-[1-(2-methylpropyl)-5-oxopyrrolidine-3-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
2-[4-(2-ethoxypyridin-3-yl)-1H-pyrazol-1-yl]-N-methylacetamide
N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1,3-dimethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N,2,5-trimethyl-N-(1H-pyrazol-5-ylmethyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-{4-[(5-cyclopentylthiophen-2-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
4-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
1-{5-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
9-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
6-methyl-5-{5-[3-(morpholin-4-yl)propyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
(2S,4R)-4-(4-{[N-(furan-2-ylmethyl)-3-methylbut-2-enamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3-(pyrrolidin-3-yl)benzamide
(3aR,6aR)-2-(2,6-difluoro-4-methoxybenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{1-[(4-ethoxyphenyl)methyl]-4-[(8-methoxy-2H-chromen-3-yl)methyl]piperazin-2-yl}ethan-1-ol
2-cyclopropyl-5-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
4-chloro-2-hydroxy-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}benzamide
5-(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonyl}-4-methylphenyl)-2-methyl-1,3-oxazole
3-{4-[(2-chlorophenyl)methyl]-4-(ethoxycarbonyl)piperidine-1-carbonyl}pyridin-1-ium-1-olate
1-[2-({[3-(dimethylamino)-2,2-dimethylpropyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)naphthalene-1-carboxamide
N,N-diethyl-1-[1-(2-ethylbutyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
methyl[(4-phenyl-1,3-thiazol-2-yl)methyl]{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
1-cyclohexyl-N3-cyclopropyl-N5-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-tert-butyl-2-[6-(ethylamino)pyridazin-3-yl]benzene-1-sulfonamide
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidin-3-ol
6-{[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}-2-methyl-2,3-dihydropyridazin-3-one
ethyl 2-({2-oxo-3-phenyl-1,8-diazaspiro[4.5]decane-8-carbonyl}amino)acetate
2-chloro-4-{[3-(2-methoxybenzoyl)piperidin-1-yl]methyl}phenol
4-(2-methylphenoxy)-1-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)piperidine-4-carboxylic acid
4-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-N-(oxolan-2-ylmethyl)benzenesulfonamide
1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
5-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid