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2-(2-{[4-(6-chloropyridazin-3-yl)piperazin-1-yl]methyl}phenoxy)acetamide
1-benzyl-N3-[2-(3-chlorophenyl)ethyl]-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-methyl-N-[1-(3-methylphenyl)piperidin-4-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[4-phenyl-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]ethan-1-one
(2R)-2-{5-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]-4-phenyl-1H-imidazol-1-yl}propanamide
5-{[7-(3-methoxypropyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
8-chloro-N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-methylquinoline-4-carboxamide
(3S,4S)-1-(5-methylpyridine-3-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
4-phenyl-N-(1-{1-[1-(pyridin-2-yl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
5-methyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-ethyl-8-fluoro-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
2-(3-hydroxypiperidin-1-yl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}acetamide
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-[(1-ethyl-1H-imidazol-2-yl)methyl]-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-methyl-5-{4-[2-(oxolan-3-yl)-1H-imidazol-1-yl]phenyl}-2H-1,2,3,4-tetrazole
N'-cycloheptyl-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}butanediamide
1-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-methoxypiperidine
ethyl 4-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole-3-carboxylate
4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
4-(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}pyrrolidin-2-yl)-3,5-dimethyl-1,2-oxazole
N-[(2-chlorophenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[(3R,4S)-1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
(3aS,6aR)-5-[2-(methylsulfanyl)pyrimidin-4-yl]-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[2-({[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
(1s,4s)-4-[4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carbonyl]cyclohexan-1-ol
3-[1-(1,3-benzothiazole-2-carbonyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(4-ethylpiperazin-1-yl)-3-(2-methoxy-4-{[4-(propan-2-yl)piperazin-1-yl]methyl}phenoxy)propan-2-ol
2-(4-cyclopentyl-1,4-diazepan-1-yl)quinoline
1,5-dimethyl-2-phenyl-4-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}-2,3-dihydro-1H-pyrazol-3-one
2-{[(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-3-yl)oxy]methyl}pyridine
3-{[(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
4-{1-[5-(3-phenyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]ethyl}morpholine
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[3-(methylsulfanyl)propyl]piperidine
5-ethyl-5-(1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
2-[1-benzyl-5-(dimethylamino)-1H-1,2,4-triazol-3-yl]benzamide
3-(1H-1,3-benzodiazol-1-yl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}propanamide
8-methoxy-2-methyl-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-(dimethylamino)-2-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-2,3-dihydropyridazin-3-one
6-methyl-N4-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyrimidine-2,4-diamine
N-[(6-methylpyridin-2-yl)methyl]-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamide
4-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine
5-[1-(3-fluoropyridine-4-carbonyl)pyrrolidin-2-yl]-N-(1H-pyrazol-3-yl)thiophene-2-carboxamide
3-butyl-1-methyl-4-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}piperazin-2-one
2-[(quinolin-8-yloxy)methyl]-N-[2-(1,3-thiazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
4-{3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-6-(4-methyl-1H-pyrazol-1-yl)pyrimidine
N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]-2H-1,3-benzodioxole-5-carboxamide
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
(3S,9aR)-3-(2-methylpropyl)-8-(3-phenylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione