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N'1-benzyl-N'1-(prop-2-en-1-yl)cyclopropane-1,1-dicarboxamide
(1-{[2-(3-chlorophenyl)-6,7-dimethoxyquinolin-3-yl]methyl}piperidin-4-yl)methanol
3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[1-(propan-2-yl)piperidin-4-yl]-1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]ethan-1-one
methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl][(2E)-2-methylbut-2-en-1-yl]amine
5-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-2,1,3-benzoxadiazole
6-phenyl-2-{2-[2-(pyridin-4-yl)-1H-imidazol-1-yl]ethyl}-2,3-dihydropyridazin-3-one
3-{2-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-3-(2-oxopyrrolidin-1-yl)propanamide
1-[4-(methylamino)pyrimidin-2-yl]-4-phenoxypiperidine-4-carboxylic acid
4-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-4-oxobutanamide
N-{2-methyl-5-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]phenyl}cyclopropanecarboxamide
N-(3-methyl-1-{7-[3-(thiophen-2-yl)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)acetamide
2-methyl-5-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,4-dihydropyridin-4-one
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}acetamide
1-(3-fluorophenyl)-6,6-dimethyl-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
4-{1-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]ethyl}morpholine
5-methyl-N-(pyridin-4-ylmethyl)-4-{[1-(thiophen-2-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2-chloro-4-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}pyridine
3-[5-(5-ethylthiophene-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-N,2-dicyclopentylacetamide
(2S,4S)-4-amino-N-ethyl-1-{[6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}pyrrolidine-2-carboxamide
3-[2-(2,6-difluorophenyl)ethyl]-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
N-(3,4-difluorophenyl)-1-(quinoline-3-carbonyl)piperidin-3-amine
N-ethyl-N-methyl-2-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}acetamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,2,3-thiadiazole-4-carboxamide
methyl (2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-{[(3-methylphenyl)methyl]carbamoyl}pyrrolidine-2-carboxylate
3-[(2R,3R,6R)-5-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
6-hydroxy-N-(5-methanesulfonamido-2-methylphenyl)-1,4-oxazepane-4-carboxamide
N-cyclopropyl-N-(1-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
5-{[5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-2-(methoxymethyl)-4-methyl-1,3-thiazole
(4aS,7aR)-1-(2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}acetyl)-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{1-[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]piperidin-4-yl}-1,3-oxazolidin-2-one
2-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-1-(piperidin-1-yl)ethan-1-one
3-hydroxy-3-({[2-(1H-imidazol-4-yl)ethyl]amino}methyl)-1-[(3-methylphenyl)methyl]piperidin-2-one
1-({5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propan-2-ol
(1S,5R)-N-[3-(methylsulfanyl)phenyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-(1-benzothiophen-2-ylmethyl)-2-oxo-6-(piperidin-1-ylmethyl)-1,2-dihydropyridine-3-carboxamide
2-(methylamino)-1-[4-(2-methylphenoxy)piperidin-1-yl]ethan-1-one
1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(pyridin-3-yl)ethan-1-one
2-methoxy-N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
6-fluoro-2-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
[1-({1-[(1S,2R)-2-butylcyclopropanecarbonyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
N-{1-[4-hydroxy-2-(phenoxymethyl)pyrimidine-5-carbonyl]pyrrolidin-3-yl}acetamide
(3S,4S)-4-cyclopropyl-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidine-3-carboxylic acid
2-{4-[3-(phenoxymethyl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
2-methyl-8-{2-[4-(piperidin-3-yl)-1H-1,2,3-triazol-1-yl]ethoxy}quinoline
5-[1-(1H-indol-3-ylmethyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
3-(2-methoxyethyl)-1-(5-methylthiophene-3-carbonyl)piperidine-3-carboxylic acid