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5-(3-methoxyphenyl)-N-(morpholin-2-ylmethyl)furan-2-carboxamide
{[4-methoxy-3-(methoxymethyl)phenyl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
3-(6-chloro-2-methylpyridin-3-yl)-1-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1-(pyridin-3-ylmethyl)urea
2-(2-ethyl-1H-imidazol-1-yl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]ethan-1-one
2-(4-fluorophenyl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
methyl 2-({3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carbonyl}amino)benzoate
N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-N-cyclopentyl-5-methylthiophene-2-carboxamide
5-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-3-(2-phenylethyl)-1,2,4-oxadiazole
1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-[(1S)-1-(3-methylpyridin-2-yl)ethyl]urea
N-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
(3S)-4-{2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-1,3-dimethylpiperazin-2-one
8-{[5-(2-fluorophenyl)furan-2-yl]methyl}-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(2S)-2-[(5-methyl-1-propyl-1H-pyrazol-4-yl)formamido]-3-phenylpropanamide
5-ethyl-6-methyl-N4-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]pyrimidine-2,4-diamine
N-[1-(furan-2-carbonyl)piperidin-3-yl]-4-(pyridin-2-yl)pyrimidin-2-amine
{3-[(4-fluorophenyl)methyl]-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl}methanol
(1-methyl-1H-imidazol-2-yl)({1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl})methanol
N-[1-(2-methylpropanoyl)piperidin-3-yl]-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(5-propyl-1,2,4-oxadiazol-3-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}-2-(propan-2-yl)-1,3-oxazole
N-[3-(3-ethylphenoxy)propyl]-N-methyloxolane-3-carboxamide
2-(morpholin-2-yl)-1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]ethan-1-one
2-[2-(dimethylamino)ethyl]-8-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
5-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
2-[2-(2,4-dimethoxyphenyl)phenyl]ethan-1-amine
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(3-methyl-1,2-oxazol-5-yl)acetamide
(3aR,6aR)-2-cyclopropanecarbonyl-5-[(5-methylpyrazin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(1H-imidazol-2-yl)-N-[(4-sulfamoylphenyl)methyl]benzamide
N4-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
1-(3-chlorophenyl)-4-(2-hydroxypyridine-3-carbonyl)-5-methylpiperazin-2-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[4-(thian-4-yl)piperazin-1-yl]propan-1-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-[(3-methylthiophen-2-yl)methyl]piperidine-3-carboxamide
4-(5-methyl-1H-indol-3-yl)pyridin-2-amine
1-(2-chlorophenyl)-5-methyl-4-[3-(pyridin-4-yl)propanoyl]piperazin-2-one
2-[(3,4-difluorophenyl)methyl]-8-(3-ethoxypropanoyl)-2,8-diazaspiro[4.5]decan-3-one
3-({4-[3-(4,4-difluoropiperidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
N-(3-ethylphenyl)-2,7-diazaspiro[4.5]decane-7-carboxamide
(1S,2R)-N1-ethyl-N1-[2-(3-methoxyphenoxy)ethyl]-N2-methylcyclohexane-1,2-dicarboxamide
2-methyl-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
6-fluoro-N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-2,1,3-benzothiadiazole-4-sulfonamide
3-cyclopropyl-6-[4-(4-fluorophenyl)oxan-4-yl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
5-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}isoquinoline
7-(2-methoxyethyl)-2-[(6-methoxypyridin-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
7-cyclobutaneamido-N-(1H-indol-2-ylmethyl)-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
ethyl 8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxylate
1-{[(2S,4S)-1-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-4-fluoropyrrolidin-2-yl]methyl}-3,3-dimethylurea
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
2-({[(3R,4R)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
1-(4-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-1,4-diazepan-1-yl)ethan-1-one