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(3R)-1-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}pyrrolidin-3-ol
2-(4,6-dimethyl-1-benzofuran-3-yl)-1-[4-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]ethan-1-one
N-({1-[(3-fluoro-2,4-dimethylphenyl)methyl]piperidin-3-yl}methyl)methanesulfonamide
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoacetamide
1-(cyclopropylmethyl)-4-(1-methyl-1H-pyrazole-4-carbonyl)-2-(propan-2-yl)-1,4-diazepane
2-ethyl-N-(2-methoxy-5-methylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
6-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
6-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-1,3-benzothiazole
N-[2-(4-methoxyphenyl)ethyl]-2-[4-(6-oxo-1,6-dihydropyridazin-4-yl)piperazin-1-yl]acetamide
4-{4-[({[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]methyl}amino)methyl]phenyl}but-3-yn-1-ol
N-[1-(hydroxymethyl)cyclopentyl]-2-[(3-methoxyphenyl)amino]butanamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)acetamide
4-[(6-hydroxy-1,4-diazepan-1-yl)sulfonyl]benzoic acid
8-[2-(2,5-dimethylphenyl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
8-(butan-2-yl)-1-ethyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-benzyl-2-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}acetamide
methyl 3-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]benzoate
{6-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]pyridin-2-yl}methanol
(3S,5R)-1-(1H-pyrazole-3-carbonyl)-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
3-(3-fluorophenyl)-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)propan-1-one
1-{3-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propyl}-1H-pyrazole
2-[(furan-3-ylmethyl)(methyl)amino]-2-(4-methanesulfonylphenyl)acetic acid
1-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-(1-oxo-2,3-dihydro-1H-inden-5-yl)urea
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-(4-fluoro-3-methylphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]propanamide
5-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)-2-(trifluoromethyl)pyridine
{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
1-[1-(2-ethoxyacetyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
4-(5-methylpyridin-2-yl)-1-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]piperidin-4-ol
2-(5-{11-oxo-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-13-yl}furan-2-yl)benzonitrile
N-(2-{[3-(3-methylphenyl)-1H-pyrazol-4-yl]formamido}ethyl)pyridine-3-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-(2-methylpyrrolidin-1-yl)pyridine-3-carboxamide
N-methyl-6-phenyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[4-(pyridin-2-yl)piperazin-1-yl]-3-[1-(thiophene-2-carbonyl)piperidin-3-yl]propan-1-one
2-(2,3-dimethoxy-5-methylphenyl)-4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
3-(3-hydroxy-2,2-dimethylpropyl)-7-methyl-3H,4H-thieno[3,2-d]pyrimidin-4-one
2-[(3S,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidine-1-carbonyl]naphthalen-1-ol
N-cyclopropyl-1-[1-(1-methyl-1H-imidazole-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
5-{4-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
4-{[(furan-2-ylmethyl)(3-methylbutan-2-yl)amino]methyl}benzonitrile
1-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
(1R,9aR)-1-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-octahydro-1H-quinolizine
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1-(piperidin-1-yl)cyclohexane-1-carboxamide
4,4,4-trifluoro-1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]butan-1-one
9-methoxy-4-[(4-methoxy-3-methylphenyl)methyl]-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[2-(3-phenyl-1H-pyrazole-5-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-(4,6-dimethylquinazolin-2-yl)piperidin-4-amine