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4-[1-(3-phenylpropyl)-5-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
6-(3-{2-azabicyclo[2.2.1]heptan-2-yl}propanoyl)-N-[4-(methylsulfanyl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
3-methyl-6-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}-2,3-dihydro-1,3-benzoxazol-2-one
N2,N2-dimethyl-N5-(pyridin-4-ylmethyl)-5,6,7,8-tetrahydroquinazoline-2,5-diamine
methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})[(1-propyl-1H-imidazol-2-yl)methyl]amine
3-[(3R,4S)-1-(6-chloroquinolin-4-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
4-{3-[2-(2-methylphenyl)-1H-imidazol-1-yl]propyl}morpholine
3-(2-methoxyethyl)-7-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
2-amino-1-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-one
8-(2-chlorobenzenesulfonyl)-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
6-cyclopentyl-1-methyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S,4S)-4-cyclopropyl-1-[2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]pyrrolidine-3-carboxylic acid
4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)-1-(2-methylbutyl)piperidine
1-tert-butyl-N-[2-(4-fluorobenzenesulfonyl)ethyl]-5-oxopyrrolidine-3-carboxamide
1-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-2-(9-methyl-9H-carbazol-3-yl)ethan-1-one
2-(4-fluorophenoxy)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1-(oxolane-2-carbonyl)piperidine
5-(2,4-difluorophenoxymethyl)-N-[1-(pyridin-4-yl)propyl]-1,2-oxazole-3-carboxamide
3-(2-{1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}ethyl)phenol
(4aS,7aR)-1-[(4-ethoxyphenyl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-methyl-5-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}-3-(2-methylpropyl)-1H-pyrazole
N-[2-(1H-1,3-benzodiazole-1-carbonyl)phenyl]-3-(3-methyl-1H-1,2,4-triazol-5-yl)propanamide
2-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-fluoro-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
5-methanesulfonyl-2-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]pyrimidin-4-amine
4-methyl-3-{1H-pyrazolo[3,4-b]pyridin-1-yl}pyridine
ethyl 2-[(3-phenylprop-2-yn-1-yl)(propyl)amino]acetate
5-[1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N,N-dimethylpyrimidin-4-amine
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
(3S,4R)-1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N4,N4,5-trimethyl-N2-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-2,4-diamine
2-[3-(1-methyl-1H-pyrazol-3-yl)phenyl]-5-(trifluoromethyl)pyridine
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
2-[3-(1H-imidazol-1-yl)propyl]-9-(2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-N-(furan-2-ylmethyl)-N-methyl-5-[(quinolin-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{4-[2-(dimethyl-1,3-thiazol-4-yl)acetamido]-2-methylphenyl}pentanamide
5-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2,3-dimethylbenzene-1-sulfonamide
N-[(1S)-2-hydroxy-1-phenylethyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-(2-methanesulfonamidoethyl)-1,3-benzothiazole-6-carboxamide
ethyl 4-{6-[4-(pyrrolidin-1-yl)benzoyl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate
N-benzyl-N-(2-hydroxyethyl)-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
4-{7-[ethoxy(phenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl}-N,N-dimethylpiperidine-1-carboxamide
2-methyl-N-[(4-phenyloxan-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-acetyl-N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}benzamide
1-(2-{1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}piperidin-1-yl)ethan-1-one
2-(3,4-dichlorophenyl)-4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}morpholine
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(1-benzothiophen-2-ylmethyl)-1-benzyl-N-methylpyrrolidine-2-carboxamide
N-({1-[(6-chloropyridin-3-yl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}methyl)-2-methoxyacetamide