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4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(2,4-dimethoxy-3-methylphenyl)methyl]piperidine
8-{4-[ethyl(methyl)amino]pyrimidin-2-yl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-2,3,4-trimethoxybenzamide
1-[3-(2H-1,3-benzodioxol-5-yl)-3-phenylpropanoyl]-1,4-diazepan-5-one
2-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-N-(2-acetamidophenyl)acetamide
5-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-4-methylpyrimidine
1-[(cyclopropylcarbamoyl)methyl]-4-methanesulfonyl-1,4-diazepane-6-carboxylic acid
N-[2-(3-chlorophenyl)ethyl]-1-(2-methoxyethyl)-5-(3-methylpiperidine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
4-(3-hydroxypropanoyl)-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(3S,4R)-1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-4-phenylpyrrolidine-3-carboxylic acid
4-hydroxy-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
3-(1-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)pyridine
N-[(3-carbamoyl-1,2,4-oxadiazol-5-yl)methyl]-1-cyclohexylpiperidine-4-carboxamide
4-(5-{[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
7-(pyridin-2-yl)-4-{[4-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(3-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-3-oxopropyl)azepan-2-one
N-[2-(4-chlorophenoxy)ethyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
(4S)-3-(2-{6-oxa-9-azaspiro[4.5]decan-9-yl}-2-oxoethyl)-4-phenyl-1,3-oxazolidin-2-one
methyl 5-{5-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-{1-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]piperidin-4-yl}pyridin-2-amine
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methylpyridin-2-amine
methyl (2S)-2-{[1-cyclohexyl-5-(methylcarbamoyl)-4-oxo-1,4-dihydropyridin-3-yl]formamido}-3-phenylpropanoate
2-[(2-{[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}ethyl)amino]-6-methyl-3,4-dihydropyrimidin-4-one
2-{4-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
N,N-dimethyl-3-(1-{[4-(pyridin-3-yl)phenyl]methyl}piperidin-3-yl)propanamide
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(propan-2-yloxy)ethan-1-one
4-[(2-hydroxyethyl)sulfamoyl]-N-[2-(pyridin-4-yl)ethyl]benzamide
2-(4-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-N,N-dimethylacetamide
N-(2-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxy}propyl)imidazo[1,2-a]pyridine-2-carboxamide
(2R,3R,6R)-N-(furan-2-ylmethyl)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-2,3,4-trimethoxy-N-methylbenzamide
{3-[(2-fluorophenyl)methyl]-1-(naphthalen-1-ylmethyl)piperidin-3-yl}methanol
4-(pyridin-2-yl)-N-[2-(quinolin-8-yloxy)ethyl]pyrimidin-2-amine
N,4-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
2-(2,4-dichlorophenoxy)-N-[(3S)-piperidin-3-yl]acetamide
4-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
2,3,5-trimethyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-N-methyl-2-phenylacetamide
(3R,4R)-1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
9-[(4-chlorophenyl)methyl]-2-[3-(dimethylamino)propyl]-2,9-diazaspiro[5.5]undecan-3-one
5-[(dimethylamino)methyl]-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylfuran-2-carboxamide
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-4-hydroxy-2-methylpyrimidine-5-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-6-methyl-4-oxo-N-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
8-(2-methyl-1,3-thiazole-4-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
ethyl 3-(2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamido)propanoate
1-{2-[1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
7-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidine
4-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]-5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidine
4-(3,4-dimethylphenyl)-3-{[ethyl(methyl)amino]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one