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3-(1-methyl-1H-imidazol-2-yl)-1-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,4-dimethyl-1,3-thiazole-5-carboxamide
1-(2-methoxyphenyl)-4-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl)piperazine
(2S,4S)-N-ethyl-4-(furan-2-amido)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]pyrrolidine-2-carboxamide
1-[2-(1H-imidazol-2-yl)benzoyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]piperidin-4-ol
2-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1,4,5-trimethyl-1H-imidazole
N,N-dimethyl-2-[(1S,5R)-6-(quinoxaline-6-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[1-(4-methylphenyl)propyl]propanamide
N-(2-hydroxyethyl)-5-(1H-pyrazol-1-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)furan-2-carboxamide
6-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-2-carbonitrile
2-(4-pentamethylbenzoylpiperidine-1-carbonyl)morpholine
N-(3-cyanophenyl)-2,8-diazaspiro[4.5]decane-2-carboxamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methylpiperidine-4-carboxamide
[(2S)-1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol
(4aR,7aS)-4-(1-benzofuran-5-ylmethyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-[3-(dimethylamino)pyrazin-2-yl]-N,N-bis(propan-2-yl)benzamide
N-(1-benzothiophen-2-ylmethyl)-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-3-(1,3-dimethyl-1H-pyrazol-4-yl)urea
1-(4,7-dimethylquinazolin-2-yl)-N-(oxan-4-yl)piperidine-4-carboxamide
4-(2-methoxypyridine-3-carbonyl)-1-(4-methylphenyl)piperazin-2-one
1-{2-[({2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}ethan-1-one
2-methoxy-5-[2-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]pyridine
2-ethyl-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrimidine-5-carboxamide
4-{[(2S,4S)-4-[(4-fluorophenyl)sulfanyl]-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]methyl}quinoline
2-{[2-(2,4-difluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}-6-methoxyphenol
6-methoxy-3-[2-oxo-2-(4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)ethyl]-2,3-dihydro-1H-indol-2-one
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
1-({3-[4-(piperidin-1-yl)butoxy]phenyl}methyl)piperidine-3-carbonitrile
2-[3-(naphthalen-1-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetic acid
3-[3-(3-propyl-1,2,4-oxadiazol-5-yl)propyl]-1H-indole
(1R,5R)-6-(2H-1,3-benzodioxole-5-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)propanamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-methanesulfonamidopropanamide
[(2-methoxyphenyl)methyl][(6-methoxypyridin-3-yl)methyl]propylamine
N-[1-(1H-imidazol-1-yl)butan-2-yl]-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
2-(2-hydroxyethyl)-9-[5-(methoxymethyl)furan-2-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
6-{4-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperazin-1-yl}pyrazine-2-carboxamide
1-[4-(pyridin-4-yl)piperidin-1-yl]-2-(1H-1,2,4-triazol-3-ylsulfanyl)ethan-1-one
4-methoxy-N-[4-(4-{[2-(pyridin-4-yl)ethyl]amino}piperidin-1-yl)phenyl]benzamide
2-chloro-6-fluoro-N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]benzamide
8-chloro-2-[4-(2-ethoxyethyl)piperazine-1-carbonyl]quinoline
9-[4-(morpholine-4-carbonyl)piperazin-1-yl]-3-azaspiro[5.5]undecane
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
N-cyclobutyl-3-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}sulfonyl)benzamide
1-{2-[(butylamino)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-(2-hydroxyethyl)-4-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(4-methylpiperazin-1-yl)pyrimidine-5-carboxamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-5-phenyl-1,2-oxazole-3-carboxamide
4-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}-2-[5-(methylcarbamoyl)thiophen-2-yl]pyrrolidine-1-carboxamide