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4-({4-cyclopropyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1-(3-methylphenyl)-1H-pyrazole
2-{4-[4-(piperidin-1-ylmethyl)benzoyl]piperazin-1-yl}pyrazine
N-(1-{1-[(2-hydroxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methylbenzamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N,2,6,8-tetramethylquinoline-4-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-(thiophen-2-yl)propanamide
(3S)-N,N-dimethyl-1-(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)pyrrolidin-3-amine
3-{[3-phenyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1H-isoindol-1-one
(3R,5S)-N3-(4-fluorophenyl)-N5-(2-hydroxyethyl)-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
3-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(pentan-3-yl)-N-propylbenzamide
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N,6-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
{[3-(2-fluorophenyl)-1H-pyrazol-5-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
1-[(2-chloro-4-fluorophenyl)methyl]-N-(cyclobutylmethyl)-N-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N'-cycloheptyl-N-[(5-methylpyrazin-2-yl)methyl]butanediamide
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-ol
1-[2-(difluoromethoxy)benzoyl]-2-(3-methoxypropyl)piperidine
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-methyl-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-{[(2-hydroxyethyl)[(1-methyl-1H-imidazol-2-yl)methyl]amino]methyl}-6-methylquinolin-4-ol
6-{[(2-aminopyrimidin-5-yl)methyl](methyl)amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
3-[(4-chlorophenyl)methyl]-1-(1,4-oxazepan-6-ylmethyl)urea
3-{4-[(4-chlorophenyl)methyl]piperazine-1-carbonyl}-1,4,6-trimethyl-1,2-dihydropyridin-2-one
2-(2-methyl-1,3-thiazol-4-yl)-1-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
8-fluoro-2-[({[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}amino)methyl]quinolin-4-ol
(1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanamine
(2S,4S)-4-amino-N,N-diethyl-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]pyrrolidine-2-carboxamide
2-[1-(propan-2-yl)-4-(pyridin-2-ylmethyl)piperazin-2-yl]ethan-1-ol
N-ethyl-N-(2-methoxyethyl)-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-[4-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)morpholin-3-yl]-N,N-dimethylacetamide
N-(1-benzothiophen-2-ylmethyl)-1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]piperidin-4-amine
3-(3-methoxyphenyl)-5-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-1H-pyrazole
N-[2-(7-{[4-(diethylamino)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-4-fluorobenzamide
3-(4-fluorophenyl)-4-[3-(pyridin-4-yl)propanoyl]piperazin-2-one
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl})amine
8-fluoro-2-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-1,4-dihydroquinolin-4-one
N-{2-[(4-fluorophenyl)formamido]ethyl}-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-(1,3-dihydro-2-benzofuran-5-yl)-3-[1-(4-methoxyphenyl)-5-oxopyrrolidin-3-yl]urea
2-benzyl-4-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]morpholine
8-(2,3-dihydro-1H-inden-2-yl)-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-6-(5-methyl-1,3-oxazole-4-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(dimethyl-1,2-oxazol-4-yl)methyl]benzamide
2-(3-methoxyphenyl)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
N-[2-(2,4-dichlorophenyl)ethyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
(3R,4S)-4-cyclopropyl-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-3-amine
7-(2,2-dimethylpropyl)-2-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-2,7-diazaspiro[4.5]decane
1-[1-(5,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
1-[2-(dimethylamino)ethyl]-4-ethyl-3-[1-(piperidine-4-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N,N-dimethyl-6-phenyl-3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]pyridin-2-amine
4-methoxy-N-(3-methoxypropyl)-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}benzamide
2-(2-chlorophenyl)-N-[2-(4-hydroxyphenyl)ethyl]-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
ethyl 4-{[4-(1,3-thiazol-4-yl)phenyl]carbamoyl}piperazine-1-carboxylate