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N-tert-butyl-4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-(2-phenylethyl)-5-(4H-1,2,4-triazol-4-ylmethyl)-1H-1,2,4-triazole
6,8-dimethyl-2-{[4-(1,3-thiazol-2-yl)piperazin-1-yl]methyl}quinolin-4-ol
6-ethyl-N-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-(morpholin-4-yl)pyrimidin-4-amine
1-ethyl-N,2,5-trimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrrole-3-carboxamide
(1R,5R)-6-benzyl-3-(2,6-dimethylpyrimidine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-(2-chlorophenyl)-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}furan-2-carboxamide
2-(2H-1,3-benzodioxol-5-yloxy)-1-[(3S,4S)-3-hydroxy-4-(1,4-oxazepan-4-yl)pyrrolidin-1-yl]ethan-1-one
4-methyl-2-propyl-6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
1-{6-[3-(morpholine-4-carbonyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}azepane
N-ethyl-6-[4-fluoro-2-(trifluoromethyl)phenyl]pyridine-3-carboxamide
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-3-(1,2-oxazinan-2-yl)propanamide
4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-carboxamide
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-2-(1H-pyrazol-3-yl)pyridine
2-{2-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]propyl}-3-methylpyridine
1-(2-methoxyphenyl)-4-[2-(propan-2-ylsulfanyl)acetyl]piperazin-2-one
6-(morpholin-4-yl)-N4-[2-(1H-1,2,3-triazol-1-yl)ethyl]pyrimidine-2,4-diamine
N-[(3R,4S)-1-[2-methyl-2-(morpholin-4-yl)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
5-(2-fluorophenoxymethyl)-N-methyl-N-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1H-pyrazole-3-carboxamide
3-phenyl-1-(1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)prop-2-yn-1-one
(3S)-1-(1-benzyl-4-phenylpiperidine-4-carbonyl)pyrrolidin-3-amine
1-methoxy-8-{2-[4-(methylsulfanyl)phenyl]acetyl}-1,8-diazaspiro[4.5]decan-2-one
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-[(3S,4R)-1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
7-[(3,4-dimethoxyphenyl)methyl]-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-(5-{1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1H-imidazol-2-yl}thiophen-2-yl)prop-2-yn-1-ol
2-methoxy-1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
8-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(2-chlorophenoxy)-1-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]piperidine
N,3,6-trimethyl-N-[1-(1,3-thiazol-5-yl)ethyl]-1-benzofuran-2-carboxamide
N-(2-methyl-2H-1,2,3-triazol-4-yl)-4-({methyl[1-(methylcarbamoyl)propan-2-yl]amino}methyl)benzamide
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-5-yl}urea
5-hydroxy-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyrazine-2-carboxamide
4-methyl-5-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]pyrimidine
1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
1-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-(1H-pyrazol-1-yl)butan-1-one
5-methyl-N4-[5-(morpholin-4-yl)pentyl]pyrimidine-2,4-diamine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclobutan-1-amine
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
3-(4-methoxyphenyl)-N-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
1-{2-[(4-benzylpiperazin-1-yl)methyl]-1,3-oxazole-4-carbonyl}-1,4-diazepan-5-one
1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N,5-dimethyl-N-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
2-(2,3-difluorophenyl)-1-[3-(pyrimidin-4-yl)piperidin-1-yl]ethan-1-one
4-{[4-(4-fluorophenyl)-1,4-diazepan-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
6-methoxy-N-(1,2-oxazol-3-ylmethyl)-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-{[(2-fluorophenyl)methyl](methyl)amino}ethan-1-one
(1R,5R)-3-(1-tert-butyl-1H-pyrrole-3-carbonyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(1-methyl-1H-imidazol-2-yl)-1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine
2-(4-{pyrazolo[1,5-a]pyridine-7-carbonyl}piperazin-1-yl)-1,3-benzothiazole