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N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
(1S,5R)-6-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
9-(5-hydroxypyrazine-2-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-2-yl)ethan-1-one
6-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,3-benzothiazole
N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-(pyrrolidin-1-yl)benzamide
4-methoxy-N-methyl-N-(1,2-oxazol-3-ylmethyl)-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
1-(3-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-benzyl-1-methyl-3-[2-oxo-2-(piperazin-1-yl)ethyl]-2,3-dihydro-1H-indol-2-one
N-[(1R,3R)-3-aminocyclopentyl]-3-(3-hydroxy-1,2-oxazol-5-yl)propanamide
3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}propan-1-one
ethyl 4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(2S,4R)-N-ethyl-4-{[(2-fluorophenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-methyl-N-(oxan-2-ylmethyl)-2-(propan-2-yl)pyrimidine-4-carboxamide
4-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-5-ethyl-2-methylpyrimidine
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(2-methyl-1H-pyrrole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-methyl-2-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazine-1-carbonyl}azepane
2-methoxy-N-(1-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
4-[3-(5-methylfuran-2-yl)benzoyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
1-{3-[3-(thiophen-3-yl)phenyl]-1H-pyrazol-1-yl}butan-2-ol
2-[(3-chlorophenyl)methyl]-N-(pyridin-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
4-cyclobutyl-6-methyl-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidin-2-amine
N-(3-hydroxy-2,2-dimethylpropyl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
4-{4-amino-6-[(4-methylphenyl)amino]-1,3,5-triazin-2-yl}benzonitrile
3-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-4-methoxyphenol
5-methyl-4-[4-(pyrimidin-2-yloxy)piperidin-1-yl]thieno[2,3-d]pyrimidine-6-carboxylic acid
3-[({[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}amino)methyl]pyrrolidin-3-ol
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}acetamide
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(pyridine-2-carbonyl)piperidin-3-yl]propanamide
methyl[(2-methyl-1,3-oxazol-4-yl)methyl][1-(3-methylpyridin-2-yl)propan-2-yl]amine
(1R,5S,6S)-N-methyl-3-{[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxamide
1-methyl-3-({1-[2-(2-oxocyclopentyl)acetyl]piperidin-4-yl}methyl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
8-(4-cyclopentylpyrimidin-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(2,5-dimethoxyphenyl)-1-(7-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
(3S,4S)-3-hydroxy-4-[2-(4-methoxy-3-methylphenyl)-1H-imidazol-1-yl]-1λ6-thiolane-1,1-dione
N'-(2-methoxyethyl)-N-(2-methylphenyl)-N'-(pyridin-4-ylmethyl)propanediamide
2-methyl-1-({2-oxo-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-3-yl}methyl)-1,4-diazepan-5-one
2-(4-fluorophenyl)-N-(2-{7-[(4-methoxy-2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]-4-phenylpiperidin-4-ol
1-[3-(3,4-dimethoxyphenyl)propyl]-3-[1-(propan-2-yl)-1H-pyrazol-5-yl]urea
[2-(azepan-1-yl)ethyl](ethyl){[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}amine
6-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}-1,4-oxazepan-6-ol
5-amino-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-phenyl-1H-pyrazole-3-carboxamide
N-{3-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamido]phenyl}-3-phenylpropanamide
methyl 3-({4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidine-1-carbonyl}amino)benzoate
2-(3-fluorophenyl)-8-methoxy-5-(4,4,4-trifluorobutyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
6-{2-benzyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}pyridine-3-carbonitrile
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide