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4-(piperidin-4-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(2R,3R)-1'-(5-ethyl-1,2-oxazole-3-carbonyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
(1S,5R)-3-(pyridin-2-ylmethyl)-6-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane
3-{5-[2-(thiophen-2-yl)ethyl]-1H-1,2,4-triazol-3-yl}pyridine
2-(2-hydroxyethyl)-8-{[3-(trifluoromethyl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
6-methyl-4-[2-(pyrrolidine-1-carbonyl)piperazine-1-carbonyl]-1,2-dihydroquinolin-2-one
6-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2-methyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-[3-(furan-2-yl)phenyl]-1-(morpholine-2-carbonyl)piperidine-4-carboxamide
2-methoxyethyl (1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
methyl[(3-methyl-1,2-oxazol-5-yl)methyl]{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
1-[1-(3-phenylpropyl)piperidin-4-yl]-N-[(1r,4r)-4-hydroxycyclohexyl]piperidine-4-carboxamide
9-(2,6-diaminopyrimidin-4-yl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-N-(2-phenylethyl)acetamide
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-5-methanesulfonyl-2-methylpyrimidin-4-amine
6-[(2-fluorophenyl)methoxy]-4-(2-methylpropanoyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
N-(1-acetylpiperidin-4-yl)-4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carboxamide
N-[2-(3-methoxyphenyl)ethyl]-6-[2-(thiophen-3-yl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[2-(4-cyclohexyl-1,4-diazepan-1-yl)-2-oxoethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}(thiophen-2-yl)methanol
N-benzyl-N-methyl-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
N4-[(5-methylthiophen-2-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
9-{2-[ethyl(methyl)amino]propanoyl}-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-cyclopropyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,3-oxazole-4-carboxamide
2-(ethylamino)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidine-5-carboxamide
2-[2-(azepan-1-ylmethyl)-4-(pyrimidin-2-yl)phenoxy]-N-[(3-fluorophenyl)methyl]acetamide
(1R,7S)-3-(3,4-dimethylphenyl)-N-methyl-4-oxo-N-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-{[1-(4-fluorophenyl)pyrrolidin-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
(4aR,7aS)-N,N-diethyl-4-(5-methyl-1,2-oxazole-3-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-(adamantan-1-yl)-N-methyl-N-[2-(morpholin-4-yl)propyl]acetamide
5-fluoro-3-(oxan-2-ylmethyl)-3,4-dihydroquinazolin-4-one
2-(dimethylamino)-8-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
(1R,5R)-6-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)[(2-methyl-1,3-thiazol-5-yl)methyl]amine
N-{2-[({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]ethyl}acetamide
(4aS,8aR)-1-(3-hydroxypropyl)-2-oxo-N-(2-phenylethyl)-decahydro-1,6-naphthyridine-6-carboxamide
N-(2-methylpropyl)-2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]-N-(thiophen-3-ylmethyl)acetamide
3-({[(3-chloro-4,5-diethoxyphenyl)methyl]amino}methyl)-7-fluoro-1,2-dihydroquinolin-2-one
(4aR,8aS)-6-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
4-(2,3,4-trimethoxyphenyl)pyridin-3-amine
1-methyl-4-(1-{4-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-1,2,3-triazol-1-yl}propan-2-yl)piperazine
N-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}pyrazolo[1,5-a]pyridine-7-carboxamide
N-[4-(furan-2-yl)phenyl]-1-[3-(1H-pyrazol-4-yl)propanoyl]piperidine-3-carboxamide
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]({[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
9-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[5-(oxolan-2-yl)-1,3,4-thiadiazol-2-yl]-2-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]acetamide
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(prop-2-en-1-yl)piperazine
8-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(3-phenylpropyl)-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,4-diazepane
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide