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N3-butyl-1-(furan-2-ylmethyl)-N5-[(1-hydroxycyclohexyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-4-(pyridin-2-yl)pyrimidin-2-amine
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-1H-pyrazole-3-carboxamide
N-[3-(2-methoxyphenoxy)propyl]-N,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
4-[2-amino-3-cyano-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyridin-4-yl]benzamide
N-(2-hydroxyethyl)-N-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(phenylsulfanyl)acetamide
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-1H-1,3-benzodiazole-5-carboxamide
2-({[1-(furan-3-ylmethyl)piperidin-4-yl]oxy}methyl)pyridine
7-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]butanamide
2-[(3-methoxyphenyl)methyl]-8-(pyrrolidine-1-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[(2,4-difluorophenyl)methyl]-3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
3-benzyl-8-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-1-(4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-N-(cyclohexylmethyl)piperidine-1-carboxamide
1-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-(furan-2-yl)propan-1-one
ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}){[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methylpyridin-2-yl)methyl]acetamide
6-methyl-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-3H,4H-thieno[2,3-d]pyrimidin-4-one
N3-[(4-chlorophenyl)(phenyl)methyl]-N5-ethyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(1R,5R)-6-[2-(ethylamino)pyrimidine-5-carbonyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
5-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)pyrazin-2-ol
4-{1-[6-(4-ethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidin-4-yl}pyridine
7-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-2-methyl-2,7-diazaspiro[4.5]decane
(1S,5R)-3-(3-phenylpropyl)-6-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
4-[3-(1H-imidazol-1-yl)pyrrolidine-1-carbonyl]-7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
N-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
ethyl({[2-(morpholin-4-yl)quinolin-3-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-one
9-[2-(2,5-dimethylphenyl)acetyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-2-(3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)acetamide
[(3R,4R)-1-[(5-methylfuran-2-yl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
5-{1-[(2-methoxypyrimidin-5-yl)methyl]pyrrolidin-2-yl}-N-(pyridin-3-yl)thiophene-2-carboxamide
3-({3-oxo-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-4-yl}methyl)-1λ6-thiolane-1,1-dione
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-fluorophenyl)urea
3-benzyl-8-(1H-indol-2-ylmethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(dimethylamino)-1-(4-ethoxypiperidin-1-yl)-2-(4-methylphenyl)ethan-1-one
1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
1-(3-{1-[(2-methoxyphenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)-1H-pyrazole
methyl({2-methylimidazo[1,2-a]pyridin-3-yl}methyl){[2-(propan-2-yl)pyrimidin-5-yl]methyl}amine
4-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}azetidin-3-yl)pyridine
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
4-ethyl-5-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
N-[(2-ethoxypyridin-3-yl)methyl]-2-(4-phenylpiperidin-1-yl)acetamide
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
(2R,3R)-3-amino-1'-(pyridine-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol