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3-(2-oxo-2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
2-(4-chlorophenyl)-4-(3-fluoropyridin-4-yl)morpholine
1-(cyclopropylmethyl)-N-methyl-5-[(6-methylpyridin-2-yl)methyl]-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-[5-(hydroxymethyl)furan-2-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)propane-1,2-diol
1-(2-methoxypyridin-3-yl)-3-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}urea
2-(2-chlorophenyl)-N,3-dimethyl-N-(propan-2-yl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
(3-{2-[1-(3-chloro-2-fluorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-phenylpiperazine
3-{5-[5-(methoxymethyl)thiophene-2-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyridine
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
(3S,4R)-3-benzyl-1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4-methylpiperidin-4-ol
7-methyl-2-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-[3-({[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amino}methyl)-1H-indol-1-yl]acetamide
5-methyl-N-{[3-(morpholin-4-ylmethyl)phenyl]methyl}-1,2-oxazol-3-amine
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-[3-(pyridine-2-carbonyl)piperidin-1-yl]propan-1-one
3-{[4-(2-phenylphenyl)-1H-1,2,3-triazol-1-yl]methyl}pyridine
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
(2S)-1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)pyrrolidine-2-carboxamide
3-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}pyridine
2-[3-(1H-imidazol-1-yl)pyrrolidin-1-yl]-N-[2-(4-methoxyphenyl)ethyl]acetamide
1-ethyl-1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
N,5-dimethyl-4-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
2-[(1-{[2-(dimethylamino)ethyl](methyl)amino}hex-5-en-2-yl)oxy]-5-fluoro-N,N-dimethylpyrimidin-4-amine
1-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-3-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}urea
(1R,2S)-2-[4-(3-methoxyphenyl)-3-oxopiperazine-1-carbonyl]-N-methylcyclohexane-1-carboxamide
2-methyl-6-(1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-4-yl)pyrimidin-4-ol
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methylpyridin-2-amine
7-(cyclohexylmethyl)-2-(pyridin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
5-(2-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-oxoethyl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-cyclobutyl-4-[(2-fluorophenyl)methyl]-1,4-diazepan-5-one
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N,N-diethyl-5-methyl-1H-pyrazole-4-carboxamide
2-(2-methoxypyrimidine-5-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
1-(3-fluorobenzoyl)-4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
N-[(4-fluorophenyl)methyl]-2-(3-methoxyphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[(2-fluorophenyl)methyl]piperazine
4-methyl-2-(1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
(4aS,8aR)-1-(3-hydroxypropyl)-6-[3-(1H-pyrrol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
(9aR)-8-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-(1-{[3-(benzyloxy)phenyl]methyl}piperidin-3-yl)morpholine
N-[2-({[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)ethyl]acetamide
2-(propan-2-yl)-5-(3-propoxypiperidine-1-carbonyl)-1,3-benzoxazole
2-methyl-9-(1-methyl-1H-pyrazole-3-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
5-{[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]methyl}-N-(propan-2-yl)pyrimidin-2-amine
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(oxan-2-ylmethyl)amine
3-{1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}benzoic acid
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[1-(pyridin-3-yl)propan-2-yl]amine
ethyl({[(3R,4S)-1-(2-methoxyethyl)-4-propylpyrrolidin-3-yl]sulfamoyl})methylamine
methyl (1R,3S,3aR,6aS)-3-[2-(difluoromethoxy)phenyl]-1-ethyl-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
3-{[3-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl}benzoic acid