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1-cyclopentyl-N-[(4-methoxyphenyl)methyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
ethyl 5-(1-methyl-1H-pyrazole-5-carbonyl)-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-{1-[1-(2-cyclopropylacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
1-(azepan-1-yl)-3-(3-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}phenoxy)propan-2-ol
2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)acetamide
3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(1-propylpiperidin-4-yl)propanamide
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-6-(4-fluorophenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
6-ethyl-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-2-oxo-1,2-dihydropyridine-4-carboxamide
(1R,3S)-7-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}-3-methoxy-7-azaspiro[3.5]nonan-1-ol
N-benzyl-N,7-dimethyl-6-oxo-2,7-diazaspiro[4.5]decane-2-sulfonamide
2-[1-(3-methylbut-2-en-1-yl)-4-(pyridin-3-ylmethyl)piperazin-2-yl]ethan-1-ol
N-[(3,5-difluorophenyl)methyl]-2-(dimethylamino)-2-(3-methylphenyl)acetamide
4-[({[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}amino)methyl]hepta-1,6-dien-4-ol
1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidine-3-carbonitrile
methyl 1-[(3R,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-(1-ethylpiperidin-4-yl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
5-{1-[(1-benzyl-1H-imidazol-2-yl)methyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
5-acetyl-N-[(4-methoxyphenyl)methyl]-N-(oxolan-2-ylmethyl)thiophene-3-carboxamide
N-({5-[(2,4,5-trimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[4-(3-methoxybenzoyl)piperazin-1-yl]propan-1-one
4-(2-methoxyphenoxy)-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
(1R,7S)-3-[(4-fluorophenyl)methyl]-N-methyl-4-oxo-N-(pyrazin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]amine
3-(4-methylpiperazine-1-carbonyl)-N-(2-phenylethyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(3-methoxypropyl)-8-[(1-methyl-1H-indol-3-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3,4-dimethoxyphenyl)-1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
3-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]-1H-pyrazole-5-carboxamide
1-(cyclohexylmethyl)-N5-[(2,4-dimethoxyphenyl)methyl]-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-7-(1H-inden-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4,6-dimethyl-2-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidine
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]acetamide
2-amino-4-(3,5-dimethyl-1-benzofuran-2-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
5-(6-methoxypyridin-2-yl)-1,2,3,4-tetrahydroisoquinoline
5-[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]quinoxaline
2-{1-[(3-chlorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1,3-thiazole
(4aS,8aS)-2-[3-(2-fluorophenyl)benzoyl]-decahydro-2,7-naphthyridin-4a-ol
2-hydroxy-N-{2-[2-methyl-5-(morpholine-4-sulfonyl)-1H-1,3-benzodiazol-1-yl]ethyl}propanamide
{4-[3-methyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]phenyl}methanol
ethyl 4-{[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]amino}piperidine-1-carboxylate
1-(3-methylbut-2-en-1-yl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
5-methyl-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-1,3-oxazole-4-carboxamide
2-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-9-oxa-2-azaspiro[5.5]undecane
6-[1-(thiophen-2-yl)propan-2-yl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-[2-(1,1-dioxo-1λ6-thiolan-3-yl)ethyl]-N-(propan-2-yl)benzamide
methyl 3-(2-chlorobenzamido)-5-({[3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}methyl)benzoate
2-(2-methoxypyridin-3-yl)-1,3-thiazole-4-carboxamide
2-cyclohexyl-2-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]acetic acid
1-[2-(1,1-dioxo-1λ6-thiolan-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-(naphthalen-1-ylmethyl)piperidine-3-carboxamide
(1R,5S,6R,7S)-3-(2-aminoethyl)-N-[(3-methoxyphenyl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]decane-6-carboxamide