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1-(2-ethylbutyl)-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
3-({2-[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[2-(4-chlorobenzenesulfonamido)ethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
2-{[5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-phenyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-2-(trimethyl-1H-pyrazol-1-yl)acetamide
2,3-dimethyl-5-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]benzene-1-sulfonamide
methyl 3-(4-fluorobenzenesulfonamido)-5-{[2-(1,3-thiazol-4-yl)acetamido]methyl}benzoate
1-(2-phenylethyl)-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
1-methyl-5-({2-[3-(morpholin-4-ylmethyl)phenyl]-1H-imidazol-1-yl}methyl)pyrrolidin-2-one
(3aS,6aS)-2-cyclohexyl-5-(pyrimidin-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-2-methyl-4,5,6,7-tetrahydro-2H-indazole
(2R,3R)-3-amino-1'-(2H-1,3-benzodioxole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[2-(4-chlorophenyl)morpholin-4-yl]-6-methoxypyrimidin-2-amine
2-(2-chloro-4-fluorophenyl)-1-{octahydropyrrolo[1,2-a]piperazin-2-yl}ethan-1-one
2-[(4-chlorophenyl)sulfanyl]-N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]acetamide
1-[3-(1H-pyrazol-1-yl)propyl]-4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidine
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(1,2-oxazole-3-carbonyl)piperidine
N-({1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
2-butyl-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-2,5-dihydro-1H-pyrrole
6-ethyl-4-methyl-N-[(5-methylpyrazin-2-yl)methyl]quinolin-2-amine
{3-[(2,4-difluorophenyl)methyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}methanol
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl)[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(methylsulfanyl)propan-1-one
{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(isoquinolin-5-ylmethyl)methylamine
(3S,9aR)-3-benzyl-8-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
1-cyclohexyl-4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-hydroxy-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-amino-1-[4-(2,5-dihydro-1H-pyrrol-1-yl)-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
[1-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)piperidin-2-yl]methanamine
4-(1H-imidazol-1-ylmethyl)-1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperidin-4-ol
1-methyl-4-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1H-indole
[(3-fluorophenyl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(oxolan-2-ylmethyl)amine
4-({[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]amino}methyl)benzene-1-sulfonamide
3-{2-[4-(2-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
4-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]benzene-1-sulfonamide
3-{3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl}propanamide
3-(2-methoxyethyl)-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidine-3-carboxylic acid
6-cyclobutyl-2-[4-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
4-[4-(3-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]-1-[(2E)-2-methylbut-2-en-1-yl]piperidine
{2-ethoxy-5-[1-(pentan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}methanol
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)pyridin-2-amine
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[(pyridin-3-ylmethyl)amino]methyl}piperidin-2-one
2-(1-{[1-(4-methoxycyclohexanecarbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-(4-{5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}thiophen-2-yl)ethan-1-one
1-{[2-(carboxymethoxy)-5-chlorophenyl]methyl}-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-{4-[2-(2,5-dioxoimidazolidin-1-yl)acetamido]-2-methoxyphenyl}-2,2-dimethylpropanamide
(2-{3-[3-(5-ethylpyrimidin-2-yl)phenyl]-1H-pyrazol-1-yl}ethyl)dimethylamine