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4-[(2,1,3-benzoxadiazol-5-ylmethyl)amino]-1-(3-phenylpropyl)pyrrolidin-2-one
1-(2H-1,3-benzodioxole-5-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-[2-(morpholin-4-yl)-2-oxoethyl]-4-[(4-phenylphenyl)methyl]piperazin-2-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
3,6-dimethyl-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-1-benzofuran-2-carboxamide
3-[2-(2,6-difluorophenyl)ethyl]-1-[4-(propan-2-yl)-1,2,3-thiadiazole-5-carbonyl]piperidine
N3-(2H-1,3-benzodioxol-5-ylmethyl)-N5-ethyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
(2S,4R)-N-ethyl-1-(1H-imidazol-2-ylmethyl)-4-[2-(5-methyl-1H-pyrazol-1-yl)acetamido]pyrrolidine-2-carboxamide
7-methoxy-3-({methyl[(3-methylthiophen-2-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
N3-cyclooctyl-N5-(cyclopropylmethyl)-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
6-[2-amino-4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]-2,3-dihydropyridazin-3-one
N-[(4-chlorophenyl)(pyridin-4-yl)methyl]-5-hydroxy-4-oxo-4H-pyran-2-carboxamide
1-[4-(3-chlorophenyl)piperazin-1-yl]-3-[(3S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-(dimethylamino)piperidin-3-yl]propan-1-one
methyl (1R,3S,3aR,6aS)-3-(3-ethoxy-4-hydroxyphenyl)-1-ethyl-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-methyl-5-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
N-(cyclopropylmethyl)-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1'-benzoyl-5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(3S)-3-ethyl-4-[4-(4H-1,2,4-triazol-4-yl)benzoyl]morpholine
(1S,9aR)-1-(2-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}ethyl)-octahydro-1H-quinolizine
N-({6-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]pyridin-3-yl}methyl)acetamide
(1S,6R)-9-[2-(2-acetyl-4,5-dimethoxyphenyl)acetyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
1-ethyl-N-[3-(propan-2-yloxy)propyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(4-phenylpiperazin-1-yl)-3-(1-{spiro[2.5]octane-1-carbonyl}piperidin-4-yl)propan-1-one
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[2-(4-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[1-(pyridin-4-yl)propyl]amine
5-[(4-methyl-1H-pyrazol-1-yl)methyl]-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
methyl (2S,4S,5R)-5-(2-fluorophenyl)-4-{[(2-methoxyphenyl)methyl]carbamoyl}-1-methylpyrrolidine-2-carboxylate
2-benzyl-8-(dimethyl-1,3-oxazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-{[2-(3-fluorophenyl)piperidin-1-yl]sulfonyl}morpholine
ethyl 4-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl}piperazine-1-carboxylate
1-(cyclohexylmethyl)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
1-cyclohexyl-4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-2-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-3-amine
N-(2-hydroxypropyl)-5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carboxamide
1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[2-(trifluoromethyl)phenyl]ethan-1-one
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-N-[3-(1H-pyrazol-1-yl)propyl]pyrimidin-2-amine
1-phenyl-4-(2,6,8-trimethylquinoline-4-carbonyl)piperazin-2-one
2-(dimethylamino)-1-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}-2-(4-methylphenyl)ethan-1-one
ethyl 2-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-1,3-oxazole-4-carboxylate
N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-2-(thiophene-2-sulfonamido)acetamide
2-{4-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperazin-1-yl}-1,3-benzothiazole
N-[(1-cyclohexylpyrrolidin-3-yl)methyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]-4-(1H-imidazol-1-ylmethyl)piperidine
1-[4-(4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazin-1-yl)phenyl]ethan-1-one
3-(oxolan-3-yl)-5-[5-(1H-pyrazol-1-ylmethyl)furan-2-yl]-1,2,4-oxadiazole
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-N,N-diethylpiperidine-3-carboxamide
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-1-[4-(2-methoxyphenyl)piperazin-1-yl]propan-1-one
N-[2-(dimethylamino)ethyl]-4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-ethyl-6-{4-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-1-yl}-N-methylpyrimidin-4-amine
2-amino-N,N-bis(1,3-oxazol-4-ylmethyl)-4-phenylpyrimidine-5-carboxamide