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1-(3-methylpiperidin-1-yl)-3-[4-(2-phenylethyl)piperazin-1-yl]propan-1-one
3-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-5,6-dimethyl-1,2-dihydropyridin-2-one
{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
4-{1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}-2-(propan-2-yl)pyrimidine
3-(4-ethoxy-2-fluorophenyl)-1-[1-(4-methylpyridin-2-yl)propyl]urea
N-{[5-fluoro-7-(4-fluoro-3-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-[3-(dimethylamino)-1-phenylpropyl]-4-(1H-pyrazol-3-yl)benzamide
8-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2,8-diazaspiro[4.5]decan-3-one
1,5-dimethyl-4-{[4-(naphthalen-2-yl)piperazin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
2-cyclopentyl-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
4-(4-methoxyphenyl)-6-[(3-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
6-methyl-4-[1-(3-methylphenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
3-(1-methyl-1H-imidazol-2-yl)-1-[2-(1H-pyrazol-1-yl)benzoyl]piperidine
2-(3-methoxypropyl)-8-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
1-{3-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
2-{[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]amino}pyridine-4-carboxamide
5-methyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
dimethyl({4-methyl-5-[1-(thiophene-2-sulfonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
3-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanoic acid
3-{1-[2-(1H-indazol-1-yl)acetyl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-[2-(2,5-dimethylphenoxy)ethyl]-2-(2-hydroxyphenoxy)-N-methylacetamide
2-(3-methoxyphenyl)-1-[(4-methyloxan-4-yl)methyl]azetidine
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]acetamide
8-{[1-phenyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
(1R,2S,4R)-N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
1-methyl-2-oxo-8-[(2-phenylethyl)carbamoyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(3S,4R)-1-(5-methylpyridine-3-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-methylbenzamide
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-(piperidin-3-yl)urea
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-N'-(3-ethylphenyl)butanediamide
3-(2-methylphenyl)-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}pyrrolidin-3-ol
ethyl 4-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-3-yl}piperazine-1-carboxylate
3-[4-({5-[(4-chlorophenyl)sulfanyl]furan-2-yl}methyl)piperazin-1-yl]propan-1-ol
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetamide
(1S,5R)-3-(pyrazine-2-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
N-[(3-chlorophenyl)methyl]-1-(methoxymethyl)-N-(2-methylpropyl)cyclopropane-1-carboxamide
3-{4-[1-(cyclohexylmethyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}-1λ6-thiolane-1,1-dione
4-({2-[2-(4-ethylpiperazin-1-yl)ethoxy]phenyl}methyl)thiomorpholine
N-(1-{7-[(2,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)propanamide
1-[2-methyl-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)urea
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-3-(2-methylphenyl)-3-phenylpropanamide
1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
4-(4-{1-[2-(2-chlorophenyl)ethyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-7-methyl-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-{[4-(dimethylamino)oxan-4-yl]methyl}-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
(3R,5S)-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
N-methyl-N-[2-(4-methylpiperidin-1-yl)ethyl]-5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
1-[4-(2-amino-5-ethyl-6-methylpyrimidin-4-yl)-1,4-diazepan-1-yl]-2,2,2-trifluoroethan-1-one