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(3R,5R)-N-[3-(dimethylamino)propyl]-1-(naphthalen-2-ylmethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
(3R,4R)-1-(2-hydroxy-3-methylbenzoyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)[3-(methylsulfanyl)propyl]amine
N-[4-({[3-(morpholin-4-yl)propyl]carbamoyl}methoxy)phenyl]propanamide
2-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-cyclopentyl-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propanamide
2-[1'-(3-cyclopentylpropanoyl)-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl]acetamide
N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1-(propan-2-yl)piperidine-3-carboxamide
4-{7-[2-(methylsulfanyl)pyridine-3-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}morpholine
2-[(cyclopropylmethyl)(thiophen-3-ylmethyl)amino]butan-1-ol
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-2-(morpholin-2-yl)acetamide
2-(4-methoxy-3-methylphenyl)-2-[4-(pyridin-4-yl)piperazin-1-yl]acetic acid
2-({2-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
(3R,9aR)-3-benzyl-8-(2-chlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-butyl-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
4-hydroxy-2-(phenoxymethyl)-N-[1-(thiophen-2-yl)propan-2-yl]pyrimidine-5-carboxamide
N-[1-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperidin-3-yl]acetamide
5-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}-1-phenyl-1H-1,2,3-triazole
5-(2-methanesulfonylethyl)-3-(oxan-4-yl)-1H-1,2,4-triazole
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[2-(1H-pyrazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-ethyl-9-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]sulfamoyl}-N-(oxolan-3-ylmethyl)benzamide
N-[(3R,4S)-4-cyclopropyl-1-[2-(2-methoxyethoxy)acetyl]pyrrolidin-3-yl]-1-methyl-1H-pyrazole-4-carboxamide
9-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-6,7-dimethoxy-1-methyl-1,2,3,4-tetrahydroisoquinoline
1-methyl-N-[(2-methyl-1,3-oxazol-4-yl)methyl]-N-(pyridin-3-ylmethyl)piperidin-4-amine
1-(2-chlorophenyl)-3-(1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
8-methyl-3-{8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
5-cyclopropyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
3-amino-1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
6-(cyclopentylamino)-2-methylheptan-2-ol
(3aR,6aS)-N-(6-phenoxypyridin-3-yl)-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[1-(thiophen-2-yl)propan-2-yl]propanamide
(1-{1-[1-(2-methoxyphenyl)piperidin-4-yl]piperidin-3-yl}piperidin-4-yl)methanol
1-[3-(dimethylsulfamoyl)propyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
3-ethyl-3-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-(1-methyl-1H-indazol-6-yl)urea
N-cyclopropyl-1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}piperazine-2-carboxamide
N-cyclohexyl-N-methyl-3-({[(4-methyl-1H-imidazol-5-yl)methyl]amino}methyl)pyridin-2-amine
5-ethyl-N-[2-(1-methylpiperidin-2-yl)ethyl]pyrimidin-2-amine
(1S,5R)-3-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
butyl 3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
4-(cyclohex-3-en-1-yl)-1-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1H-1,2,3-triazole
N2-[(2-aminopyridin-3-yl)methyl]-5-fluoro-N4,N4-dimethylpyrimidine-2,4-diamine
N-[(5-methylpyrazin-2-yl)methyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(1-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)methanol
5-[(2-cyclohexylpyrimidin-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(3S,4S)-1-[6-(dimethylamino)pyridine-3-carbonyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
4-{5-[(2S)-1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine