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methyl 5-[(1-acetylpiperidin-4-yl)amino]-3-(4-methoxybenzamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(1-methyl-1H-pyrazol-4-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]propan-1-one
N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(morpholin-4-yl)-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
4-(4-chlorophenyl)-1-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]butan-1-one
N-(3-methoxypropyl)-N-{[2-(3-methylphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}oxolane-2-carboxamide
1,6-dimethyl-3-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
1-[7-(1-benzothiophen-3-yl)-9-[2-(pyridin-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
2-{4-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
methyl 3-(7-chloro-2-{[(1-methylcyclopropyl)formamido]methyl}-2,3-dihydro-1-benzofuran-5-yl)benzoate
N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-[(dipropylamino)methyl]benzamide
N-cyclohexyl-3-{[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]sulfamoyl}benzamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
3-(2-fluorophenyl)-3-(2-{4-[(3-fluorophenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-1-methylpyrrolidine-2,5-dione
(2S)-2-amino-3-(4-hydroxyphenyl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
1-[2-(2-methylpropanesulfonyl)ethyl]-2-[4-(methylsulfanyl)phenyl]-1H-imidazole
2-(morpholin-2-yl)-1-(2-phenylpyrrolidin-1-yl)ethan-1-one
(2R,3R,6R)-5-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-3-(4H-1,2,4-triazol-4-yl)propanamide
3-{3-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-4,6-dimethyl-1,2-dihydropyridin-2-one
dimethyl[1-(3-{1-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-1H-imidazol-2-yl}phenyl)ethyl]amine
N-[(2-methoxyphenyl)methyl]-N-propyl-1H-indole-5-carboxamide
2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetic acid
1-(4-methylphenyl)-3-{2-[1-(oxan-4-yl)piperidin-3-yl]ethyl}urea
1'-{[3-(morpholin-4-yl)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]methylamine
3-methyl-5-(2-{8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}ethyl)-1,2-oxazole
2-(pyridin-2-ylmethyl)-9-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(2-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-4-methoxyphenoxy)-2-hydroxypropyl]piperidin-4-ol
(1R,9S)-5-amino-12-methyl-3-[2-(prop-2-en-1-yloxy)phenyl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
(3S,4R)-1-[4-(4-fluorophenyl)oxane-4-carbonyl]-N,N-dimethyl-4-propylpyrrolidin-3-amine
N-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
2-(cyclohex-1-en-1-yl)-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
N-[1-({[2-(2-methyl-1H-indol-1-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]pyridine-2-carboxamide
2-{1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}-6-methyl-1H-1,3-benzodiazole
N,N,4-trimethyl-6-(4-{[1-(1-methyl-1H-pyrazol-4-yl)propyl]amino}piperidin-1-yl)pyrimidin-2-amine
N-cyclobutyl-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
methyl 1-(naphthalen-2-ylmethoxy)-2-oxo-8-(quinolin-5-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
2-(cyclopropylmethyl)-9-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]pyridin-4-amine
1-[4-(1H-pyrazol-1-yl)benzoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-{[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
6-methyl-2-oxo-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]-1,2-dihydropyridine-4-carboxamide
8-[2-(4-fluorophenoxy)acetyl]-2-phenyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-(aminomethyl)-4-(2-ethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(2-fluorophenyl)ethan-1-one
N-cyclopentyl-4-(1-methyl-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(oxolan-2-ylmethyl)-1-(propan-2-yl)-N-(thiophen-3-ylmethyl)piperidine-4-carboxamide