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6-(cyclopropylmethoxy)-4-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}piperidin-2-one
5-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]-1,2-dihydropyridin-2-one
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
[1-(oxane-4-carbonyl)-3-propylpiperidin-3-yl]methanol
3-({[cyclopropyl(pyridin-2-yl)methyl](methyl)amino}methyl)-6-methyl-1,2-dihydroquinolin-2-one
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
1-(2-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)azepan-2-one
N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-{2-[1-(3-hydroxy-2,2-dimethylpropyl)-1H-imidazol-2-yl]quinolin-6-yl}acetamide
4-[(benzylsulfamoyl)(methyl)amino]butanoic acid
3-({[(3-chlorophenyl)methyl]amino}methyl)-1-[(2-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
3-{2-[3-(2-hydroxyethoxy)phenyl]-1H-imidazol-1-yl}-N,4-dimethylbenzamide
ethyl 4-(4-{2-[(oxolan-2-ylmethyl)carbamoyl]ethyl}piperidin-1-yl)piperidine-1-carboxylate
methyl 5-[(2,3-dihydro-1,4-benzodioxin-6-yl)carbamoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2,2-dimethyl-N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]propanamide
N-(4-{4-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]piperidin-1-yl}phenyl)-2,4-dimethylbenzamide
1-[3-({4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)phenyl]ethan-1-one
2-[(4-butanoyl-6-hydroxy-1,4-diazepan-1-yl)methyl]benzonitrile
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-({7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}sulfanyl)acetamide
5-methanesulfonyl-1'-(3-methylpyrazin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-ethyl-N-[(4-methoxyphenyl)methyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
3-(2-methylphenyl)-3-[2-oxo-2-(4-propylpiperazin-1-yl)ethyl]-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
(3aR,6aR)-2-cyclopropanecarbonyl-N-[(3-methylpyridin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-ethyl-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-5-methylthiophene-3-carboxamide
N-[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]-2-methyl-3-[(pyridin-2-ylmethyl)amino]benzamide
N-[(4,6-dimethylpyridin-3-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
methyl({1-[1-(3,5,5-trimethylhexyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)amine
{4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
(4aR,7aS)-1-(2-methoxyacetyl)-4-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-methyl-5-(morpholine-4-carbonyl)-1-(2-phenylethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
6-(4-chlorophenyl)-N-(1H-1,2,4-triazol-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-(oxane-2-carbonyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
ethyl 2-{[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)carbamoyl]amino}acetate
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(4-fluorobenzoyl)pyrrolidin-3-yl]methanol
N-cyclopentyl-N-{[3,5-dimethoxy-4-(oxolan-2-ylmethoxy)phenyl]methyl}-5-methylthiophene-2-carboxamide
4-ethyl-6-{4-[(4-methanesulfonylphenyl)methyl]piperazin-1-yl}pyrimidine
1-(2-propyl-1,3-thiazole-4-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
4-methyl-2-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)phenol
N-(2-{7-[(2,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
5-fluoro-2-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
1-{4-[(3-methylbutyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
1-{2-oxo-2-[2-oxo-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-3-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]urea
3-methyl-8-(4-phenyl-1H-imidazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4-phenyl-N-{1-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
3-{2-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one